SCHEMBL7435254

SCHEMBL7435254

CCC(CC)CCCC(N)Oc1ccncc1NC(=O)c1c[nH]c2c1C(=O)CCC2

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 4/20 0.33
DHODH Q02127 2/20 0.33
BUB1 O43683 3/20 0.33
GSK3B P49841 7/20 0.32
MAPT P10636 3/20 0.32
ATR Q13535 1/20 0.32
EHMT2 Q96KQ7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7433522 0.88 GSK3A (0.34) GSK3ADHODHBUB1GSK3BMAPT
SCHEMBL7435249 0.83 BUB1 (0.35) GSK3ABUB1GSK3BMAPTATR
SCHEMBL7392263 0.81 GSK3B (0.46) GSK3ABUB1GSK3BMAPTATR
SCHEMBL6095690 0.81 BUB1 (0.36) GSK3ABUB1GSK3BMAPTATR
SCHEMBL7439659 0.80 GSK3B (0.33) GSK3ADHODHBUB1GSK3BMAPT
SCHEMBL6093224 0.80 ATR (0.37) GSK3ABUB1GSK3BMAPTATR
SCHEMBL7392028 0.80 GSK3B (0.45) GSK3ABUB1GSK3BMAPTATR
SCHEMBL8051137 0.78 GSK3B (0.45) GSK3ABUB1GSK3BMAPTATR
SCHEMBL6093811 0.77 ATR (0.46) GSK3ABUB1GSK3BMAPTATR
SCHEMBL6093421 0.77 BUB1 (0.39) GSK3ADHODHBUB1GSK3BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1210328-A1 FUSED PYRROLECARBOXAMIDES: A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2002-06-05 EP disclosed
WO-2001016103-A1 FUSED PYRROLECARBOXAMIDES: GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2001-03-08 WO disclosed