SCHEMBL7439659

SCHEMBL7439659

CCC(CC)CC(CCN)(CC(CC)CC)Oc1ccncc1NC(=O)c1c[nH]c2c1C(=O)CCC2

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 6/20 0.33
MAPT P10636 2/20 0.33
BUB1 O43683 2/20 0.32
GSK3A P49840 2/20 0.32
PIM3 Q86V86 5/20 0.31
PIM2 Q9P1W9 5/20 0.31
PIM1 P11309 5/20 0.31
DHODH Q02127 1/20 0.31
ATR Q13535 2/20 0.30
RXFP1 Q9HBX9 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7450644 0.89 PIM1 (0.34) GSK3BMAPTBUB1GSK3APIM3
SCHEMBL7439920 0.88 PIM3 (0.33) GSK3BMAPTBUB1PIM3PIM2
SCHEMBL7392263 0.82 GSK3B (0.46) GSK3BMAPTBUB1GSK3AATR
SCHEMBL7435254 0.80 GSK3A (0.33) GSK3BMAPTBUB1GSK3ADHODH
SCHEMBL7435249 0.80 BUB1 (0.35) GSK3BMAPTBUB1GSK3APIM3
SCHEMBL7392028 0.79 GSK3B (0.45) GSK3BMAPTBUB1GSK3AATR
SCHEMBL6095690 0.79 BUB1 (0.36) GSK3BMAPTBUB1GSK3APIM3
SCHEMBL6093224 0.78 ATR (0.37) GSK3BMAPTBUB1GSK3APIM3
SCHEMBL8051137 0.78 GSK3B (0.45) GSK3BMAPTBUB1GSK3AATR
SCHEMBL6093719 0.77 SGMS2 (0.37) GSK3BMAPTBUB1GSK3ARXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1210328-A1 FUSED PYRROLECARBOXAMIDES: A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2002-06-05 EP disclosed
WO-2001016103-A1 FUSED PYRROLECARBOXAMIDES: GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 2001-03-08 WO disclosed