SCHEMBL7435508

SCHEMBL7435508

CCC(Cc1ccc(F)cc1)c1cc(O)c(C(CC)c2cccs2)c(=O)o1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.36
TP53 P04637 2/20 0.33
CYP2C9 P11712 1/20 0.33
LMNA P02545 3/20 0.32
TSHR P16473 1/20 0.32
POLB P06746 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32
RAB9A P51151 2/20 0.31
HPGD P15428 1/20 0.31
NPC1 O15118 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ABL1 P00519 1/20 0.31
MME P08473 1/20 0.31
CNR2 P34972 1/20 0.31
GPR55 Q9Y2T6 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7437926 0.92 ESR1 (0.39) NQO1CYP2C9POLBALDH1A1HPGD
SCHEMBL7441300 0.92 NQO1 (0.41) NQO1CYP2C9LMNATSHRPOLB
SCHEMBL7447834 0.91 NQO1 (0.37) NQO1TP53CYP2C9LMNAPOLB
SCHEMBL7443023 0.91 NQO1 (0.37) NQO1CYP2C9LMNAPOLBMEN1
SCHEMBL7435905 0.90 NQO1 (0.35) NQO1CYP2C9
SCHEMBL7439255 0.90 MAPT (0.37) NQO1TP53CYP2C9LMNAPOLB
SCHEMBL7440406 0.90 NQO1 (0.33) NQO1TP53CYP2C9TSHRMEN1
SCHEMBL7473129 0.88 MAPT (0.38) NQO1TP53TSHRPOLBMEN1
SCHEMBL7440515 0.86 NQO1 (0.40) NQO1CYP2C9LMNAPOLBMEN1
SCHEMBL7444897 0.86 NQO1 (0.36) NQO1CYP2C9POLBALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed