SCHEMBL7444897

SCHEMBL7444897

CCC(Cc1ccsc1)c1cc(O)c(C(CC)c2cccs2)c(=O)o1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.36
CYP2C9 P11712 1/20 0.33
DRD2 P14416 1/20 0.31
DRD3 P35462 1/20 0.31
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7441300 0.90 NQO1 (0.41) NQO1CYP2C9ALDH1A1POLBMAPT
SCHEMBL7437926 0.88 ESR1 (0.39) NQO1CYP2C9ALDH1A1POLBMAPT
SCHEMBL7447834 0.87 NQO1 (0.37) NQO1CYP2C9ALDH1A1POLBMAPT
SCHEMBL7443023 0.87 NQO1 (0.37) NQO1CYP2C9ALDH1A1POLBMAPT
SCHEMBL7440515 0.86 NQO1 (0.40) NQO1CYP2C9POLBMAPT
SCHEMBL7435508 0.86 NQO1 (0.36) NQO1CYP2C9ALDH1A1POLBHPGD
SCHEMBL7439255 0.86 MAPT (0.37) NQO1CYP2C9ALDH1A1POLBMAPT
SCHEMBL7480489 0.86 NQO1 (0.34) NQO1ALDH1A1POLBMAPTHPGD
SCHEMBL7444017 0.85 CYP2C9 (0.31) CYP2C9
SCHEMBL7440443 0.85 NQO1 (0.36) NQO1CYP2C9ALDH1A1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed