SCHEMBL7440406

SCHEMBL7440406

CCC(c1cccs1)c1c(O)cc(C(Cc2ccc(F)cc2)CC2CC2)oc1=O

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TAS2R14 Q9NYV8 1/20 0.31
TSHR P16473 1/20 0.31
TP53 P04637 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7451071 0.93 NQO1 (0.34) NQO1CYP2C9
SCHEMBL7440329 0.92 NQO1 (0.33) NQO1CYP2C9
SCHEMBL7437094 0.92 NQO1 (0.33) NQO1MEN1KMT2ATP53CYP2C9
SCHEMBL9281720 0.91 CNR1 (0.34) NQO1
SCHEMBL7440164 0.91 CNR1 (0.34) NQO1
SCHEMBL7443597 0.91 MAPT (0.34) NQO1MEN1KMT2ATP53CYP2C9
SCHEMBL7435508 0.90 NQO1 (0.36) NQO1MEN1KMT2ATSHRTP53
SCHEMBL7443735 0.90 TP53 (0.35) NQO1MEN1KMT2ATP53CYP2C9
SCHEMBL7444883 0.87 NQO1 (0.33) NQO1MEN1KMT2ATAS2R14TSHR
SCHEMBL7448278 0.86

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed