SCHEMBL7435559

SCHEMBL7435559

CC(C)c1ccc(-c2cc(C(C)C)ccc2O)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.55
PTGS1 P23219 1/20 0.55
CACNA1C Q13936 1/20 0.55
ALDH1A1 P00352 3/20 0.53
HTT P42858 3/20 0.53
ALOX12 P18054 2/20 0.53
GAA P10253 2/20 0.53
HIF1A Q16665 1/20 0.53
TYR P14679 3/20 0.50
RNASEH1 O60930 1/20 0.50
PTPN5 P54829 1/20 0.49
LMNA P02545 3/20 0.47
GPR35 Q9HC97 1/20 0.46
RXRA P19793 1/20 0.43
NR4A2 P43354 1/20 0.43
MAPT P10636 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
USP2 O75604 1/20 0.42
KDM4E B2RXH2 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25906319 0.90 TRPA1 (0.55) TRPA1PTGS1CACNA1CALDH1A1HTT
SCHEMBL14252297 0.90 TYR (0.48) TRPA1PTGS1CACNA1CALDH1A1HTT
SCHEMBL17707900 0.89 TYR (0.50) TRPA1PTGS1CACNA1CALDH1A1HTT
SCHEMBL22888342 0.89 PTGS1 (0.48) TRPA1PTGS1CACNA1CALDH1A1HTT
SCHEMBL4282140 0.88 PTPN5 (0.57) TRPA1PTGS1CACNA1CALDH1A1HTT
SCHEMBL11651790 0.87 TRPA1 (0.64) TRPA1PTGS1CACNA1CALDH1A1HTT
SCHEMBL23754720 0.86 BACE1 (0.46) TRPA1PTGS1CACNA1CALDH1A1HTT
SCHEMBL25898933 0.85 PTGS1 (0.57) TRPA1PTGS1CACNA1CALDH1A1HTT
SCHEMBL5951050 0.85 TYR (0.44) TRPA1PTGS1CACNA1CALDH1A1HTT
SCHEMBL14877648 0.85 TRPA1 (0.48) TRPA1PTGS1CACNA1CALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183239-A1 AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR G.D. SEARLE & CO. (US) 2002-03-06 EP disclosed
WO-2000069821-A1 AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR G.D. SEARLE & CO. (US) 2000-11-23 WO disclosed