SCHEMBL7435778

SCHEMBL7435778

CCCNC(=O)c1nc[nH]c1N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 6/20 0.42
GABRB3 P28472 6/20 0.42
GABRA2 P47869 6/20 0.42
GABRA5 P31644 1/20 0.42
GABRA3 P34903 1/20 0.42
POLB P06746 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
GAA P10253 2/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
KMT2A Q03164 1/20 0.40
MAPT P10636 2/20 0.39
LMNA P02545 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPC1 O15118 1/20 0.39
ADRB2 P07550 1/20 0.39
HSP90AA1 P07900 1/20 0.39
XBP1 P17861 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19018643 0.80 GAA (0.51) POLBTDP1GAAALDH1A1KDM4E
SCHEMBL9576486 0.77 SMN1; SMN2 (0.46) TDP1GAAALDH1A1KDM4EKMT2A
SCHEMBL9576447 0.75 SMN1; SMN2 (0.45) POLBTDP1GAAALDH1A1KMT2A
SCHEMBL13847664 0.73 NPSR1 (0.45) POLBTDP1GAAALDH1A1KDM4E
SCHEMBL15185777 0.73 KDM4E (0.43) GABRG2GABRB3GABRA2GABRA5GABRA3
SCHEMBL3536595 0.72 GAA (0.37) POLBTDP1GAAMAPTL3MBTL1
SCHEMBL13176680 0.72
SCHEMBL3258892 0.72 GDA (0.43) POLBTDP1GAAALDH1A1KDM4E
SCHEMBL1560676 0.72 GDA (0.41) POLBTDP1GAAALDH1A1KDM4E
SCHEMBL311900 0.71 KDM4E (0.64) POLBGAAALDH1A1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647227-A1 PURINONE ANTIANGINAL AGENTS. PFIZER LTD (GB) 1995-04-12 EP disclosed
WO-1994000453-A1 PURINONE ANTIANGINAL AGENTS PFIZER LIMITED (GB) 1994-01-06 WO disclosed