SCHEMBL311900

SCHEMBL311900

CCOC(=O)c1nc[nH]c1N

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.64
SMN1; SMN2 Q16637 1/20 0.56
ALDH1A1 P00352 8/20 0.51
KMT2A Q03164 5/20 0.50
MEN1 O00255 4/20 0.50
MAPK1 P28482 1/20 0.50
LMNA P02545 2/20 0.49
GAA P10253 1/20 0.49
POLB P06746 1/20 0.49
RXFP1 Q9HBX9 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CYP1A2 P05177 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2114938 0.82 KDM4E (0.63) KDM4ESMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL5433655 0.82 NPSR1 (0.46) KDM4ESMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL1417913 0.81 KDM4E (0.81) KDM4ESMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL16296266 0.80 KDM4E (0.69) KDM4ESMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL19659065 0.80 KDM4E (0.56) KDM4ESMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL10278987 0.79 KDM4E (0.59) KDM4ESMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL4957306 0.79 KDM4E (0.59) KDM4ESMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL5870445 0.78 KDM4E (0.58) KDM4ESMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL10570426 0.78 KDM4E (1.00) KDM4ESMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL5185328 0.78 KDM4E (0.77) KDM4ESMN1; SMN2ALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 107 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260098041-A1 FUSED BICYCLIC PYRIMIDONES AS WRN INHIBITORS INCYTE CORPORATION (US) 2026-04-09 US disclosed
US-12486234-B2 PAPD5 inhibitors and methods of use thereof CHILDREN'S MEDICAL CENTER CORPORATION (US) 2025-12-02 US disclosed
CN-119798159-A PAPD5 inhibitors and methods of use thereof 儿童医学中心公司 2025-04-11 CN disclosed
US-12012414-B1 Imidazo[1,5-a]pyrido[4,3-e]pyrimidines as CK2 inhibitors King Faisal University (SA) 2024-06-18 US disclosed
CN-114106000-B Imidazo [4,5-d ] pyrimidinone tricyclic derivative and antitumor application thereof 中国科学院新疆理化技术研究所 2023-11-24 CN disclosed
US-20230295166-A1 ATR INHIBITORS AND USES THEREOF ANTENGENE DISCOVERY LIMITED (CN) 2023-09-21 US disclosed
US-20230295166-A1 ATR INHIBITORS AND USES THEREOF ANTENGENE DISCOVERY LIMITED (CN) 2023-09-21 US disclosed
US-20230295166-A1 ATR INHIBITORS AND USES THEREOF ANTENGENE DISCOVERY LIMITED (CN) 2023-09-21 US disclosed
CN-116507337-A ATR inhibitors and uses thereof 上海德琪医药科技有限公司 2023-07-28 CN disclosed
EP-4192836-A1 ATR INHIBITORS AND USES THEREOF ANTENGENE DISCOVERY LIMITED (CN) 2023-06-14 EP disclosed
US-20060217387-A1 Acetylenyl-pyrazolo-pyrimidine derivatives F. HOFFMANN-LA ROCHE AG, A SWISS COMPANY (CH) 2006-09-28 US disclosed
WO-2005037257-A2 NOVEL ALANYL-AMINO PEPTIDASE INHIBITORS FOR FUNCTIONALLY INFLUENCING DIFFERENT CELLS AND TREATING IMMUNOLOGICAL, INFLAMMATORY, NEURONAL, AND OTHER DISEASES IMTM GMBH (DE) 2005-04-28 WO disclosed
WO-1992013451-A1 IMIDAZOLE PESTICIDES SCHERING AGROCHEMICALS LIMITED (GB) 1992-08-20 WO disclosed
EP-0183848-B1 POLYAZAHETEROCYCLIC DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITION Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1990-09-12 EP disclosed
US-4918074-A CALCIUM ANTAGONISTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1990-04-17 US disclosed
EP-0252682-A2 Tetrazines MAY & BAKER LIMITED (GB) 1988-01-13 EP disclosed
EP-0217142-A2 A polyazaheterocyclic compound Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1987-04-08 EP disclosed
EP-0183848-A1 POLYAZAHETEROCYCLIC DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITION Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1986-06-11 EP disclosed
US-4236005-A ANTIANXIETY AMERICAN CYANAMID COMPANY (US) 1980-11-25 US disclosed
US-4178449-A Pyrazolo[1,5-a]pyrimidines and imidazo-[1,5-a]pyrimidines AMERICAN CYANAMID COMPANY (US) 1979-12-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060217387-A1 Acetylenyl-pyrazolo-pyrimidine derivatives NAT1, TPMT, ACAT1 KDM4E 1335/4885SMN1; SMN2 831/4885ALDH1A1 90/4885
US-20260098041-A1 FUSED BICYCLIC PYRIMIDONES AS WRN INHIBITORS WRN, POLR1A, REV1 KDM4E 4779/4885SMN1; SMN2 1169/4885ALDH1A1 1354/4885
US-12486234-B2 PAPD5 inhibitors and methods of use thereof POT1, PARP15, TERT KDM4E 2610/4885SMN1; SMN2 2702/4885ALDH1A1 2425/4885
US-20230295166-A1 ATR INHIBITORS AND USES THEREOF ATR, CHEK1, CHEK2 KDM4E 2648/4885SMN1; SMN2 1298/4885ALDH1A1 4462/4885
US-12012414-B1 Imidazo[1,5-a]pyrido[4,3-e]pyrimidines as CK2 inhibitors CDK2, CSNK1A1, CSNK2A1 KDM4E 2122/4885SMN1; SMN2 1927/4885ALDH1A1 3763/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.