SCHEMBL7435853

SCHEMBL7435853

COC(=O)CCC(N)C(=O)C(CCC(=O)OC)CCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A1 P43005 1/20 0.48
CA12 O43570 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
LNPEP Q9UIQ6 2/20 0.42
ERAP2 Q6P179 1/20 0.42
SLC7A5 Q01650 1/20 0.42
METAP2 P50579 1/20 0.42
METAP1 P53582 1/20 0.42
GRIK1 P39086 1/20 0.42
MMP2 P08253 1/20 0.41
MMP3 P08254 1/20 0.41
CTSC P53634 1/20 0.41
TSHR P16473 1/20 0.41
LTA4H P09960 1/20 0.41
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7447993 0.85 SLC1A1 (0.44) SLC1A1CA12CA7CA9CA14
SCHEMBL8700502 0.84 CA12 (0.51) SLC1A1CA12CA7CA9CA14
SCHEMBL5494852 0.82 SLC7A5 (0.51) SLC1A1KDM4EALDH1A1LMNASLC7A5
SCHEMBL5934204 0.77 CA12 (0.52) CA12CA7CA9CA14KDM4E
SCHEMBL7435848 0.76 CYP2D6 (0.51) CA12CA7CA9CA14KDM4E
Phenylalanine SCHEMBL27597013 0.76 SLC7A5 (0.65) SLC1A1SLC7A5LTA4H
SCHEMBL17375358 0.76 LTA4H (0.54) SLC1A1KDM4EALDH1A1LMNASLC7A5
SCHEMBL12869912 0.76 LTA4H (0.54) SLC1A1KDM4EALDH1A1LMNASLC7A5
SCHEMBL15466662 0.75 CA12 (0.50) SLC1A1CA12CA7CA9CA14
SCHEMBL15466661 0.75 CA12 (0.50) SLC1A1CA12CA7CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5096925-A N-substituted butyramide derivatives CIBA-GEIGY CORPORATION (US) 1992-03-17 US disclosed
US-4939261-A ANALGESICS, ANTIDEPRESSANTS, HYPOTENSIVE AGENTS, NEUROLEPTIC AGENTS CIBA-GEIGY CORPORATION (US) 1990-07-03 US disclosed
EP-0185079-B1 N-SUBSTITUTED BUTYRAMIDE DERIVATIVES CIBA-GEIGY AG (CH) 1988-10-19 EP disclosed
EP-0185079-A1 CIBA GEIGY AG 1986-06-25 EP disclosed
WO-1986000066-A1 N-SUBSTITUTED BUTYRAMIDE DERIVATIVES CIBA-GEIGY AG (CH) 1986-01-03 WO disclosed