SCHEMBL7436005

SCHEMBL7436005

CCCc1cc(-c2ccccc2)nnc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 3/20 0.46
CTSK P43235 1/20 0.41
SREBF2 Q12772 1/20 0.40
SMARCA2 P51531 1/20 0.40
SMARCA4 P51532 1/20 0.40
PBRM1 Q86U86 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
MEN1 O00255 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
KMT2A Q03164 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
GABRA1 P14867 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL581419 0.86 CASP1 (0.53) CASP1SMARCA2SMARCA4PBRM1SMN1; SMN2
SCHEMBL7255679 0.83 CASP1 (0.50) CASP1SMARCA2SMARCA4PBRM1SMN1; SMN2
SCHEMBL1752936 0.83 CASP1 (0.46) CASP1SMARCA2SMARCA4PBRM1SMN1; SMN2
SCHEMBL7435124 0.83 CYP2A6 (0.44) MEN1ALDH1A1KMT2AKDM4EMAPT
SCHEMBL1752896 0.81 CASP1 (0.44) CASP1SMARCA2SMARCA4PBRM1SMN1; SMN2
SCHEMBL1752940 0.79 CASP1 (0.45) CASP1SMARCA2SMARCA4PBRM1SMN1; SMN2
SCHEMBL1752842 0.78 CASP1 (0.47) CASP1SMARCA2SMARCA4PBRM1SMN1; SMN2
SCHEMBL7438450 0.76 MAPT (0.40) CTSKSREBF2SMARCA2SMARCA4PBRM1
SCHEMBL1752910 0.76 CASP1 (0.43) CASP1SMARCA2SMARCA4PBRM1SMN1; SMN2
SCHEMBL1753114 0.75 NPC1 (0.47) CASP1SREBF2SMN1; SMN2MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5278161-A Racemic mixtures HOFFMANN-LA ROCHE INC. (US) 1994-01-11 US disclosed
EP-0464572-A2 Aminoacid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1992-01-08 EP disclosed