SCHEMBL7436009

SCHEMBL7436009

O=C(O)C(Br)c1cccc(C(F)(F)F)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.55
ACP3 P15309 2/20 0.55
PNMT P11086 1/20 0.51
IDO1 P14902 1/20 0.49
TDO2 P48775 1/20 0.49
PPARG P37231 4/20 0.48
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
SRD5A2 P31213 1/20 0.46
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
AKR1C3 P42330 1/20 0.46
AKR1C2 P52895 1/20 0.46
EPHX1 P07099 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
POLB P06746 1/20 0.46
CYP3A4 P08684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015679 1.00 CES2 (0.55) CES2ACP3PNMTIDO1TDO2
SCHEMBL29099863 0.86 CES2 (0.53) CES2ACP3PNMTIDO1TDO2
SCHEMBL7469419 0.86 PNMT (0.53) CES2ACP3PNMTIDO1TDO2
SCHEMBL330908 0.86 CES2 (0.53) CES2ACP3PNMTIDO1TDO2
SCHEMBL10454464 0.85 CES2 (0.51) CES2ACP3PNMTIDO1TDO2
SCHEMBL18952889 0.84 CES2 (0.57) CES2ACP3PNMTIDO1TDO2
SCHEMBL3312220 0.83 CES2 (0.47) CES2IDO1TDO2AKR1C3AKR1C2
SCHEMBL1760926 0.82 CES2 (0.49) CES2ACP3PNMTIDO1TDO2
SCHEMBL30523034 0.82 CES2 (0.49) CES2ACP3PNMTIDO1TDO2
SCHEMBL14176566 0.82 CES2 (0.49) CES2ACP3PNMTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110092782-B Benzo-hexaazacyclo compound and preparation method and application thereof 中国科学院广州生物医药与健康研究院 2022-10-21 CN disclosed
CN-111057024-A Sydneone and sydneone imine compound and preparation method and application thereof 华东理工大学 2020-04-24 CN disclosed
EP-1077701-A4 ANTI-VIRAL COMPOUNDS LILLY CO ELI (US) 2002-03-20 EP disclosed
US-6358971-B1 FOR INHIBITING THE GROWTH OF A PICORNAVIRUS ELI LILLY AND COMPANY 2002-03-19 US disclosed
EP-1077701-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 2001-02-28 EP disclosed
WO-1999059587-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 1999-11-25 WO disclosed
EP-0482080-B1 SMALL CYCLIC PLATELET AGGREGATION INHIBITORS GENENTECH INC (US) 1997-03-26 EP disclosed
EP-0555328-A1 PLATELET AGGREGATION INHIBITORS GENENTECH, INC. (US) 1993-08-18 EP disclosed
WO-1992007870-A1 PLATELET AGGREGATION INHIBITORS GENENTECH, INC. (US) 1992-05-14 WO disclosed
US-4260620-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1981-04-07 US disclosed
US-4202901-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1980-05-13 US disclosed
US-4197302-A HYPOTENSIVE AGENTS, 5-ETHERIFIED, ALSO ESTERS, AMIDES, HYDRAZIDES CIBA-GEIGY CORPORATION (US) 1980-04-08 US disclosed