SCHEMBL9502308

SCHEMBL9502308

O=c1c2[nH]c(Nc3ccccc3)nc2n(CC2CC2)c(=O)n1CC1CC1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 10/20 0.58
PDE4B Q07343 10/20 0.58
PDE4C Q08493 10/20 0.58
PDE4D Q08499 10/20 0.58
PDE5A O76074 9/20 0.58
LMNA P02545 1/20 0.55
GAA P10253 1/20 0.55
HTT P42858 1/20 0.55
GFER P55789 1/20 0.55
TAAR1 Q96RJ0 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
ADORA1 P30542 6/20 0.48
ADORA2A P29274 3/20 0.48
ADORA2B P29275 3/20 0.48
PCK1 P35558 3/20 0.46
ADORA3 P0DMS8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13986119 0.84 PDE4A (0.56) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7393964 0.82 PDE4A (0.54) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL13986122 0.80 PDE4A (0.66) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL13986185 0.80 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7396195 0.80 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7502502 0.78 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7436271 0.77 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7395750 0.75 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7397877 0.74 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL7397416 0.73 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DPDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0550559-A1 XANTHINES Beecham Group p.l.c. (GB) 1993-07-14 EP claimed
EP-0550559-A1 XANTHINES Beecham Group p.l.c. (GB) 1993-07-14 EP disclosed