SCHEMBL7436310

SCHEMBL7436310

CC(C)(C)OC(=O)NC(Cc1cccc(OCc2ccccc2)c1)C(=O)NC1CCCCC1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.51
CTSK P43235 5/20 0.51
CTSB P07858 4/20 0.51
BCL2 P10415 1/20 0.50
SCN9A Q15858 2/20 0.49
YAP1 P46937 2/20 0.49
CACNA1B Q00975 1/20 0.49
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
ALDH1A1 P00352 1/20 0.48
CTSL P07711 2/20 0.48
PTPN1 P18031 1/20 0.48
KDM4E B2RXH2 1/20 0.48
MME P08473 1/20 0.48
ACE P12821 1/20 0.48
CPA1 P15085 1/20 0.48
ACE2 Q9BYF1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7436304 1.00 CTSS (0.51) CTSSCTSKCTSBBCL2SCN9A
SCHEMBL7361331 0.91 BCL2 (0.61) CTSSCTSKCTSBBCL2SCN9A
SCHEMBL8552202 0.85 BCL2 (0.48) CTSSCTSKCTSBBCL2SCN9A
Ammonia Solution, Strong SCHEMBL27493136 0.84 BCL2 (0.47) CTSSCTSKCTSBBCL2SCN9A
SCHEMBL4650144 0.83 PTPN1 (0.64) CTSSCTSKCTSBBCL2YAP1
SCHEMBL31407708 0.83 PTPN1 (0.64) CTSSCTSKCTSBBCL2YAP1
SCHEMBL2552297 0.83 PTPN1 (0.64) CTSSCTSKCTSBBCL2YAP1
SCHEMBL7367771 0.83 BCL2 (0.60) CTSSCTSKCTSBBCL2SCN9A
SCHEMBL2353801 0.81 KLK5 (0.59) CTSSCTSKCTSBBCL2YAP1
SCHEMBL20905733 0.81 PTPN1 (0.55) CTSSCTSKCTSBBCL2CACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4873253-A Phenylalanine derivative and proteinase inhibitor Okamoto, Shosuke (JP) 1989-10-10 US disclosed
EP-0284632-A1 Phenylalanine derivative and proteinase inhibitor Okamoto, Shosuke (JP) 1988-10-05 EP disclosed