SCHEMBL7436627

SCHEMBL7436627

Cc1cc2ccc(C#N)cc2o1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.47
PGR P06401 6/20 0.42
MEN1 O00255 2/20 0.41
GLA P06280 2/20 0.41
KMT2A Q03164 2/20 0.41
MIF P14174 1/20 0.40
CA9 Q16790 1/20 0.40
ALDH1A1 P00352 1/20 0.40
IDO1 P14902 1/20 0.40
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
XDH P47989 1/20 0.38
SLC22A12 Q96S37 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
CSNK1D P48730 1/20 0.38
CSNK1G2 P78368 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL177345 0.85 CYP2A6 (0.52) CYP2A6PGRALDH1A1IDO1NOS3
SCHEMBL6211730 0.81 HSD17B3 (0.36) PGRMEN1GLAKMT2AMIF
SCHEMBL17401006 0.78 CYP2A6 (0.48) CYP2A6PGRMEN1GLAKMT2A
SCHEMBL11550694 0.78 CYP2A6 (0.60) CYP2A6PGRMEN1GLAKMT2A
SCHEMBL5034778 0.76 CYP2A6 (0.46) CYP2A6PGRMEN1GLAKMT2A
SCHEMBL5028054 0.76 CYP2A6 (0.46) CYP2A6PGRMIFCA9
SCHEMBL8718369 0.74 MIF (0.49) MEN1GLAKMT2AMIFCA9
SCHEMBL15842472 0.74 MIF (0.71) CYP2A6PGRMEN1GLAKMT2A
SCHEMBL9431131 0.73 PGR (0.63) CYP2A6PGRMEN1GLAKMT2A
SCHEMBL18585563 0.73 CYP2A6 (0.43) CYP2A6PGRMEN1GLAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0918768-B1 AROMATIC AMIDINE DERIVATIVES USEFUL AS SELECTIVE THROMBIN INHIBITORS C & C RES LAB (KR) 2002-01-09 EP disclosed
US-6201006-B1 ANTICOAGULANTS C & C RESEARCH LABORATORIES (KR) 2001-03-13 US disclosed
EP-0918768-A1 AROMATIC AMIDINE DERIVATIVES USEFUL AS SELECTIVE THROMBIN INHIBITORS C & C Research Laboratories (KR) 1999-06-02 EP disclosed
WO-1997045424-A1 AROMATIC AMIDINE DERIVATIVES USEFUL AS SELECTIVE THROMBIN INHIBITORS C & C RESEARCH LABORATORIES (KR) 1997-12-04 WO disclosed