SCHEMBL7436644

SCHEMBL7436644

CC(C)(C)OC(=O)CC(N)C(=O)C(C(=O)OCc1ccccc1)n1nnc(-c2cccc3ccccc23)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
SLC7A5 Q01650 1/20 0.35
LTA4H P09960 3/20 0.33
ABCG2 Q9UNQ0 2/20 0.33
SYK P43405 1/20 0.33
TDP1 Q9NUW8 2/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
MAPT P10636 1/20 0.32
XBP1 P17861 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
THRB P10828 1/20 0.31
CASP1 P29466 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7434047 0.88 CYP1A2 (0.36) CYP1A2CYP2C9CYP2C19SLC7A5LTA4H
SCHEMBL7438701 0.87 CYP1A2 (0.48) CYP1A2CYP2C9CYP2C19SLC7A5LTA4H
SCHEMBL7445782 0.86 CYP1A2 (0.35) CYP1A2CYP2C9CYP2C19SLC7A5LTA4H
SCHEMBL7431022 0.85 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19LTA4HTDP1
SCHEMBL7443562 0.85 CYP2C9 (0.36) CYP1A2CYP2C9CYP2C19SLC7A5LTA4H
SCHEMBL7441643 0.84 CCKAR (0.34) SLC7A5LTA4HTDP1ALDH1A1SMN1; SMN2
SCHEMBL7439049 0.84 CYP1A2 (0.36) CYP1A2CYP2C9CYP2C19SLC7A5LTA4H
SCHEMBL7437714 0.84 CYP1A2 (0.43) CYP1A2CYP2C9CYP2C19SLC7A5LTA4H
SCHEMBL7442267 0.83 SMN1; SMN2 (0.46) CYP1A2CYP2C9CYP2C19SLC7A5LTA4H
SCHEMBL7438488 0.83 CYP2C9 (0.34) CYP1A2CYP2C9CYP2C19SLC7A5LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710153-A INTERLEUKIN CONVERTING ENZYME INHIBITORS ONO PHRAMACEUTICAL CO., LTD. (JP) 1998-01-20 US disclosed
EP-0761680-A2 Tetrazole compounds having Interleukin-1beta converting enzyme inhibitory activity ONO PHARMACEUTICAL CO., LTD. (JP) 1997-03-12 EP disclosed