SCHEMBL7438488

SCHEMBL7438488

Cc1ccc(Cl)c(-c2nnn(C(C(=O)OCc3ccccc3)C(=O)C(N)CC(=O)OC(C)(C)C)n2)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
PTGER1 P34995 2/20 0.34
SLC7A5 Q01650 1/20 0.33
TDP1 Q9NUW8 3/20 0.33
ALDH1A1 P00352 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
L3MBTL1 Q9Y468 3/20 0.32
LTA4H P09960 3/20 0.32
MAPT P10636 2/20 0.32
THRB P10828 2/20 0.32
SYK P43405 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPY1R P25929 1/20 0.32
MAOB P27338 1/20 0.32
ADORA2A P29274 1/20 0.32
RECQL P46063 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7443562 0.86 CYP2C9 (0.36) CYP2C9CYP1A2CYP2C19PTGER1SLC7A5
SCHEMBL7433464 0.86 MAP3K5 (0.33) CYP2C9CYP1A2CYP2C19PTGER1SLC7A5
SCHEMBL7438701 0.85 CYP1A2 (0.48) CYP2C9CYP1A2CYP2C19SLC7A5TDP1
SCHEMBL7434047 0.84 CYP1A2 (0.36) CYP2C9CYP1A2CYP2C19SLC7A5TDP1
SCHEMBL7431022 0.83 CYP1A2 (0.47) CYP2C9CYP1A2CYP2C19TDP1ALDH1A1
SCHEMBL7436644 0.83 CYP1A2 (0.35) CYP2C9CYP1A2CYP2C19SLC7A5TDP1
SCHEMBL7445782 0.82 CYP1A2 (0.35) CYP2C9CYP1A2CYP2C19SLC7A5TDP1
SCHEMBL7437714 0.82 CYP1A2 (0.43) CYP2C9CYP1A2CYP2C19SLC7A5TDP1
SCHEMBL7442267 0.81 SMN1; SMN2 (0.46) CYP2C9CYP1A2CYP2C19PTGER1SLC7A5
SCHEMBL7439049 0.80 CYP1A2 (0.36) CYP2C9CYP1A2CYP2C19SLC7A5TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710153-A INTERLEUKIN CONVERTING ENZYME INHIBITORS ONO PHRAMACEUTICAL CO., LTD. (JP) 1998-01-20 US disclosed
EP-0761680-A2 Tetrazole compounds having Interleukin-1beta converting enzyme inhibitory activity ONO PHARMACEUTICAL CO., LTD. (JP) 1997-03-12 EP disclosed