SCHEMBL7436776

SCHEMBL7436776

O=C(c1cccnc1)c1c[nH]c(=O)[nH]1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.54
ALDH1A1 P00352 3/20 0.47
APP P05067 1/20 0.47
GAA P10253 1/20 0.47
HCAR3 P49019 1/20 0.47
HCAR2 Q8TDS4 1/20 0.47
F7 P08709 1/20 0.46
F3 P13726 1/20 0.46
SARM1 Q6SZW1 1/20 0.46
SIRT2 Q8IXJ6 1/20 0.46
SIRT6 Q8N6T7 1/20 0.46
SIRT1 Q96EB6 1/20 0.46
SIRT3 Q9NTG7 1/20 0.46
SIRT5 Q9NXA8 1/20 0.46
SIRT4 Q9Y6E7 1/20 0.46
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
PLOD2 O00469 1/20 0.41
PIM1 P11309 1/20 0.41
PIM3 Q86V86 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9787353 0.83 MAP2K1 (0.52) MAP2K1ALDH1A1APPGAAHCAR3
SCHEMBL7437748 0.80 PDE3B (0.46) ALDH1A1GAALMNACYP1A2CYP3A4
SCHEMBL7487387 0.80 ALDH1A1 (0.48) ALDH1A1GAAHDAC6CYP1A2CYP3A4
SCHEMBL9312864 0.76 MAP2K1 (0.54) MAP2K1ALDH1A1APPGAAHCAR3
SCHEMBL1141370 0.76 MAP2K1 (0.54) MAP2K1ALDH1A1APPGAAHCAR3
SCHEMBL29915528 0.75 ALDH1A1 (0.71) MAP2K1ALDH1A1APPGAAHCAR3
SCHEMBL1242243 0.75 ALDH1A1 (0.71) MAP2K1ALDH1A1APPGAAHCAR3
SCHEMBL9786683 0.75 NAMPT (0.59) ALDH1A1GAALMNAHIF1AHPGD
Hydrochloric Acid SCHEMBL27841975 0.73 ALDH1A1 (0.68) MAP2K1ALDH1A1APPGAAHCAR3
Thymine SCHEMBL19057050 0.72 F7 (0.58) ALDH1A1APPGAAHCAR3HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0170214-B1 THE PREPARATION OF 1,3-DIHYDRO-4-PYRIDOYL-2H-IMIDAZOL-2-ONES MERRELL DOW PHARMACEUTICALS INC. (US) 1989-09-13 EP disclosed
EP-0170214-A1 The preparation of 1,3-Dihydro-4-pyridoyl-2H-imidazol-2-ones MERRELL DOW PHARMACEUTICALS INC. (US) 1986-02-05 EP disclosed
US-4405628-A 4-Pyridylimidazolones and method of use MERRELL DOW PHARMACEUTICALS INC. (US) 1983-09-20 US disclosed
EP-0059948-A1 Novel aroylimidazolones MERRELL DOW PHARMACEUTICALS INC. (US) 1982-09-15 EP disclosed