SCHEMBL7437647

SCHEMBL7437647

O=CC1COc2cc(Cl)c(Cl)cc2O1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.44
FFAR1 O14842 5/20 0.36
FLT1 P17948 1/20 0.33
AHR P35869 1/20 0.33
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30
HPGD P15428 2/20 0.30
ALDH1A1 P00352 1/20 0.30
KMT2A Q03164 1/20 0.30
CA1 P00915 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7444491 0.89 CA2 (0.40) CA2FFAR1ALDH1A1KMT2A
SCHEMBL7434309 0.81 CA2 (0.48) CA2FFAR1AHRCA1
SCHEMBL2487394 0.81 CA2 (0.48) CA2FFAR1AHRCA1
SCHEMBL7443159 0.81 CA2 (0.48) CA2FFAR1AHRCA1
SCHEMBL7446435 0.80 AHR (0.37) AHR
SCHEMBL7434642 0.76
SCHEMBL7436292 0.74 CA2 (0.48) CA2FFAR1KMT2A
SCHEMBL7437340 0.74 CA2 (0.42) CA2KMT2A
SCHEMBL1299611 0.73 NISCH (0.44) CA2HPGDALDH1A1
SCHEMBL1299583 0.73 NISCH (0.44) CA2HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4558129-A Benzodioxanyl-hydroxyethylene-piperazinyl acetanilides which effect calcium entry and β-blockade SYNTEX (U.S.A.) INC. (US) 1985-12-10 US disclosed
US-4499100-A CARDIOUVASCULAR DISORDERS SYNTEX (U.S.A.) INC. (US) 1985-02-12 US disclosed