SCHEMBL7437758

SCHEMBL7437758

CCc1cc(N(C)c2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n2nc(SC)nc2n1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.33
ALDH1A1 P00352 4/20 0.33
HPGD P15428 4/20 0.33
HSD17B10 Q99714 2/20 0.33
UBE2M P61081 1/20 0.33
DCUN1D1 Q96GG9 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
AGTR1 P30556 3/20 0.30
AGTR2 P50052 3/20 0.30
ABCB1 P08183 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7442286 0.89 SMN1; SMN2 (0.39) HSD17B10SMN1; SMN2AGTR1AGTR2
SCHEMBL7442728 0.89 AGTR1 (0.30) SMN1; SMN2AGTR1AGTR2
SCHEMBL7446270 0.88 BRD4 (0.32) KDM4E
SCHEMBL7442350 0.85 AGTR1 (0.31) AGTR1AGTR2
SCHEMBL7446015 0.83 TSHR (0.39) KDM4EALDH1A1UBE2MDCUN1D1MAPT
SCHEMBL7439152 0.82 CRHR1 (0.33) HSD17B10AGTR1AGTR2
SCHEMBL7436578 0.81 SMN1; SMN2 (0.31) SMN1; SMN2AGTR1AGTR2
SCHEMBL7440006 0.81 ABCB1 (0.35) KDM4EALDH1A1HPGDSMN1; SMN2MAPT
SCHEMBL7444478 0.81 CRHR1 (0.37) AGTR1
SCHEMBL7433989 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed