SCHEMBL7437816

SCHEMBL7437816

CCCCNc1ncccc1C(=O)OC

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.59
HPGD P15428 2/20 0.59
KDM4E B2RXH2 2/20 0.59
HSD17B10 Q99714 1/20 0.59
RIPK1 Q13546 1/20 0.52
BDKRB1 P46663 2/20 0.48
CNR2 P34972 1/20 0.48
TLR8 Q9NR97 2/20 0.47
TLR7 Q9NYK1 2/20 0.47
LMNA P02545 1/20 0.47
RAB9A P51151 1/20 0.46
POLB P06746 1/20 0.46
HTT P42858 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
PKM P14618 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
KMT2A Q03164 1/20 0.45
MAPK8 P45983 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4771680 0.91 KDM4E (0.71) ALDH1A1HPGDKDM4EHSD17B10BDKRB1
SCHEMBL6605329 0.89 HTT (0.60) ALDH1A1HPGDKDM4EHSD17B10LMNA
SCHEMBL15635912 0.85 KDM4E (0.62) ALDH1A1HPGDKDM4EHSD17B10TLR8
SCHEMBL11492008 0.85 KDM4E (0.54) ALDH1A1HPGDKDM4EHSD17B10BDKRB1
SCHEMBL11604657 0.82 ALDH1A1 (0.46) ALDH1A1HPGDKDM4EHSD17B10RIPK1
SCHEMBL27874325 0.81 KDM4E (0.61) ALDH1A1HPGDKDM4EHSD17B10TLR8
SCHEMBL9239004 0.81 KDM4E (0.61) ALDH1A1HPGDKDM4EHSD17B10LMNA
SCHEMBL6612663 0.80 ALDH1A1 (0.68) ALDH1A1HPGDKDM4EHSD17B10LMNA
SCHEMBL14155843 0.79 ALDH1A1 (0.43) ALDH1A1HPGDKDM4EHSD17B10RIPK1
SCHEMBL7737872 0.79 KMT2A (0.49) ALDH1A1HPGDKDM4EHSD17B10POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458636-B1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them KYOWA HAKKO KOGYO KK (JP) 1995-07-12 EP disclosed
US-5248684-A CERTAIN 2-OXO-QUINOLINE CARBOXYLATES OR CORRESPONDING CARBOXAMIDES USEFUL AS ANTI-EMETICS AND SUPPRESSANTS OF MIGRAINE KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-09-28 US disclosed
EP-0458636-A1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them KYOWA HAKKO KOGYO CO., LTD (JP) 1991-11-27 EP disclosed