SCHEMBL7438146

SCHEMBL7438146

C=CC[C@@H](N)c1ccccc1-c1ccc(C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1LG2 Q9BQ51 2/20 0.40
CD274 Q9NZQ7 2/20 0.40
CA12 O43570 2/20 0.36
CA2 P00918 2/20 0.36
CA9 Q16790 2/20 0.36
CA1 P00915 1/20 0.36
KDM4E B2RXH2 3/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
POLB P06746 1/20 0.33
MMP9 P14780 1/20 0.33
SYK P43405 1/20 0.33
RAB9A P51151 5/20 0.33
NPC1 O15118 3/20 0.33
CYP2C19 P33261 1/20 0.33
LMNA P02545 2/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2474135 1.00 PDCD1LG2 (0.40) PDCD1LG2CD274CA12CA2CA9
Hydrochloric Acid SCHEMBL2480213 0.85 PDCD1LG2 (0.39) PDCD1LG2CD274CA12CA2CA9
SCHEMBL2471466 0.84 PTGS2 (0.38) PDCD1LG2CD274CA12CA2CA9
SCHEMBL2474504 0.80 ALOX5AP (0.38) PDCD1LG2CD274MAPTTP53
SCHEMBL2480866 0.79 HDAC4 (0.42) PDCD1LG2CD274KDM4ESLC6A2SLC6A3
SCHEMBL2474346 0.79 PDCD1LG2 (0.36) PDCD1LG2CD274
SCHEMBL2476054 0.77 FEN1 (0.40) MEN1KMT2ACYP2C19LMNAMAPT
SCHEMBL8995483 0.76 ESR1 (0.41) PDCD1LG2CD274CYP2C19ALDH1A1SLC6A2
SCHEMBL3105786 0.76 PTPRC (0.37) PDCD1LG2CD274CYP2C19
SCHEMBL2476954 0.76 PDCD1LG2 (0.36) PDCD1LG2CD274KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5229381-A Inhibitors of leukocyte enzyme elastase MERCK & CO., INC. (US) 1993-07-20 US disclosed
EP-0481671-A1 New substituted azetidinones as anti-inflammatory and antidegenerative agents MERCK & CO. INC. (US) 1992-04-22 EP disclosed