SCHEMBL2476954

SCHEMBL2476954

C=CCC(N)c1ccccc1-c1ccoc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1LG2 Q9BQ51 2/20 0.36
CD274 Q9NZQ7 2/20 0.36
IMPDH2 P12268 2/20 0.35
NAT1 P18440 3/20 0.34
ALDH1A1 P00352 3/20 0.33
HSD17B10 Q99714 3/20 0.33
CYP2C19 P33261 3/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
CLK4 Q9HAZ1 2/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
KMT2A Q03164 1/20 0.33
CSNK2A1 P68400 1/20 0.33
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2480213 0.80 PDCD1LG2 (0.39) PDCD1LG2CD274ALDH1A1HSD17B10CYP2C19
SCHEMBL2471466 0.76 PTGS2 (0.38) PDCD1LG2CD274ALDH1A1CYP2C19CLK4
SCHEMBL7438146 0.76 PDCD1LG2 (0.40) PDCD1LG2CD274ALDH1A1CYP2C19MEN1
SCHEMBL2474135 0.76 PDCD1LG2 (0.40) PDCD1LG2CD274ALDH1A1CYP2C19MEN1
SCHEMBL2480866 0.73 HDAC4 (0.42) PDCD1LG2CD274CYP1A2KDM4EADORA2A
SCHEMBL3105786 0.73 PTPRC (0.37) PDCD1LG2CD274CYP2C19CYP3A4ADRA1D
SCHEMBL2478616 0.72 PDCD1LG2 (0.40) PDCD1LG2CD274CYP2C19
SCHEMBL2473298 0.72 PDCD1LG2 (0.44) PDCD1LG2CD274ALDH1A1CYP2C19CYP1A2
SCHEMBL2477497 0.72 PDCD1LG2 (0.39) PDCD1LG2CD274ALDH1A1CYP2C19MEN1
Hydrochloric Acid SCHEMBL2476971 0.70 PDCD1LG2 (0.34) PDCD1LG2CD274ALDH1A1HSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2159216-B1 3-BUTENYL-1-AMINE DERIVATIVES AND THEIR USE AS Ih MODULORS FOR THE TREATMENT OF PSYCHIATIRC DISORDERS ORGANON NV (NL) 2011-10-12 EP disclosed
EP-2159216-A1 Ih - Modulators N.V. Organon (NL) 2010-03-03 EP disclosed
US-20040229910-A1 Therapeutic compounds N.V. ORGANON (NL) 2004-11-18 US disclosed
US-20020037885-A1 Therapeutic compounds DIJCKS FREDERICUS ANTONIUS (NL) 2002-03-28 US disclosed
US-6313139-B1 ADMINISTERING BENZYLAMINE DERIVATIVE FOR THERAPY OF PSYCHIATRIC DISORDER IN MAMMALS AKZO NOBEL N. V. (NL) 2001-11-06 US disclosed
US-6080773-A USEFUL FOR TREATMENT OF DEPRESSION, ANXIETY OR PSYCHOSIS AKZO NOBEL, N.V. (NL) 2000-06-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040229910-A1 Therapeutic compounds BDNF, PNMT, SLC18A2 PDCD1LG2 3624/4885CD274 2894/4885IMPDH2 2386/4885
US-20020037885-A1 Therapeutic compounds BDNF, PNMT, SLC18A2 PDCD1LG2 3624/4885CD274 2894/4885IMPDH2 2386/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.