SCHEMBL7438560

SCHEMBL7438560

CC(C)CC(C(=O)N(C)C#N)c1cc(-c2ccccc2)ccc1OC1CCN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 10/20 0.46
CTSS P25774 1/20 0.45
CTSK P43235 1/20 0.45
PIK3CD O00329 4/20 0.41
PIK3CA P42336 2/20 0.41
PIK3CB P42338 2/20 0.41
PIK3CG P48736 2/20 0.41
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38
TBK1 Q9UHD2 2/20 0.38
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
PDE4B Q07343 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4717337 0.85 CTSK (0.52) USP30CTSSCTSK
SCHEMBL4711972 0.82 CTSK (0.49) USP30CTSSCTSKPIK3CDPIK3CA
SCHEMBL4714872 0.81 CTSS (0.43) USP30CTSSCTSKPIK3CDPIK3CA
SCHEMBL4715916 0.80 CTSK (0.55) USP30CTSSCTSK
SCHEMBL4716533 0.78 CTSK (0.52) USP30CTSSCTSKPRMT5WDR77
SCHEMBL7504106 0.75 USP30 (0.43) USP30CTSSCTSKPIK3CDPIK3CA
SCHEMBL4717334 0.74 CTSK (0.70) CTSSCTSK
SCHEMBL4711970 0.72 CTSK (0.67) CTSSCTSK
SCHEMBL4714869 0.71 CTSK (0.59) CTSSCTSK
SCHEMBL6217327 0.70 CTSK (0.46) CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001049288-A9 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2001-10-25 WO disclosed