SCHEMBL7438697

SCHEMBL7438697

COC(=O)[C@@H]1NC(=O)[C@H]1CCCNC(=NC(=O)OCc1ccccc1)NC(=O)OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
HTT P42858 1/20 0.39
TPSAB1 Q15661 3/20 0.38
KEAP1 Q14145 2/20 0.38
NFE2L2 Q16236 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
MAPT P10636 1/20 0.37
TGM2 P21980 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CPB1 P15086 1/20 0.36
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
POLB P06746 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7521279 1.00 IDO1 (0.41) IDO1TDO2HTTTPSAB1KEAP1
SCHEMBL7438694 1.00 IDO1 (0.41) IDO1TDO2HTTTPSAB1KEAP1
SCHEMBL13302789 0.94 IDO1 (0.42) IDO1TDO2HTTTPSAB1KEAP1
SCHEMBL7413013 0.92 IDO1 (0.43) IDO1TDO2HTTTPSAB1KEAP1
SCHEMBL7384409 0.92 IDO1 (0.43) IDO1TDO2HTTTPSAB1KEAP1
SCHEMBL7412436 0.92 IDO1 (0.43) IDO1TDO2HTTTPSAB1KEAP1
SCHEMBL7412445 0.92 IDO1 (0.43) IDO1TDO2HTTTPSAB1KEAP1
SCHEMBL7384402 0.92 IDO1 (0.43) IDO1TDO2HTTTPSAB1KEAP1
SCHEMBL7412431 0.92 IDO1 (0.43) IDO1TDO2HTTTPSAB1KEAP1
SCHEMBL7319986 0.84 CTSK (0.46) IDO1TDO2HTTTPSAB1KEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175283-A Enzyme inhibitors for antitrypsin or antithrombin as anticoagulants BRISTOL-MYERS SQUIBB COMPANY (US) 1992-12-29 US claimed
US-5326863-A Antithrombin and antitrypsin activity BRISTOL-MYERS SQUIBB COMPANY (US) 1994-07-05 US disclosed
US-5250677-A Anticoagulants BRISTOL-MYERS SQUIBB COMPANY (US) 1993-10-05 US disclosed
US-5037819-A Anticoagulant; treating pancreatitis BRISTOL-MYERS SQUIBB COMPANY (US) 1991-08-06 US disclosed