SCHEMBL7438985

SCHEMBL7438985

CCCCC(NCC(CC(C)C)NC(=O)COc1cccc(OC)c1)C(=O)CSCc1ccco1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.40
HPGD P15428 6/20 0.40
POLB P06746 5/20 0.40
MAPT P10636 5/20 0.40
USP2 O75604 3/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
HSD17B10 Q99714 2/20 0.37
HAVCR2 Q8TDQ0 1/20 0.36
CYP2C19 P33261 3/20 0.36
CYP2C9 P11712 1/20 0.36
RECQL P46063 1/20 0.36
MAPK1 P28482 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
ALOX5 P09917 1/20 0.34
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
TSHR P16473 1/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7306946 0.93 ALDH1A1 (0.41) ALDH1A1HPGDPOLBMAPTUSP2
SCHEMBL7314560 0.93 ALDH1A1 (0.40) ALDH1A1HPGDPOLBMAPTUSP2
SCHEMBL7439502 0.92 ALDH1A1 (0.39) ALDH1A1HPGDPOLBMAPTUSP2
SCHEMBL7438981 0.89 POLB (0.40) ALDH1A1HPGDPOLBMAPTUSP2
SCHEMBL7438992 0.89 POLB (0.40) ALDH1A1HPGDPOLBMAPTUSP2
SCHEMBL7445067 0.88 ALDH1A1 (0.41) ALDH1A1HPGDPOLBMAPTUSP2
SCHEMBL7436028 0.88 ALDH1A1 (0.41) ALDH1A1HPGDPOLBMAPTUSP2
SCHEMBL7309694 0.88 HPGD (0.44) ALDH1A1HPGDPOLBMAPTUSP2
SCHEMBL7306407 0.86 POLB (0.51) ALDH1A1HPGDPOLBMAPTUSP2
SCHEMBL7310960 0.85 ALDH1A1 (0.42) ALDH1A1HPGDPOLBMAPTUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed