SCHEMBL7438987

SCHEMBL7438987

COC(C)(OC)OC(=O)N[C@@H](Cc1cnc[nH]1)C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 3/20 0.54
ICAM1 P05362 3/20 0.54
ITGAL P20701 3/20 0.54
CA1 P00915 3/20 0.48
CA2 P00918 3/20 0.48
SLC6A5 Q9Y345 1/20 0.48
CYP3A4 P08684 2/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47
SLC7A5 Q01650 1/20 0.46
SLC15A2 Q16348 1/20 0.44
HRH3 Q9Y5N1 3/20 0.44
REN P00797 2/20 0.44
CPB2 Q96IY4 1/20 0.43
MME P08473 1/20 0.43
ECE1 P42892 1/20 0.43
EPHX2 P34913 1/20 0.42
AGTR2 P50052 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1133307 0.89 ITGB2 (0.57) ITGB2ICAM1ITGALCA1CA2
SCHEMBL1132649 0.89 ITGB2 (0.57) ITGB2ICAM1ITGALCA1CA2
SCHEMBL14028689 0.89 ITGB2 (0.57) ITGB2ICAM1ITGALCA1CA2
SCHEMBL28684251 0.88 ITGB2 (0.56) ITGB2ICAM1ITGALCA1CA2
SCHEMBL6806998 0.86 ITGB2 (0.62) ITGB2ICAM1ITGALCA1CA2
SCHEMBL1486141 0.81 REN (0.49) ITGB2ICAM1ITGALHRH3REN
SCHEMBL18814494 0.81 REN (0.49) ITGB2ICAM1ITGALHRH3REN
SCHEMBL28386295 0.80 ITGB2 (0.60) ITGB2ICAM1ITGALCA1CA2
SCHEMBL18878768 0.79 REN (0.49) ITGB2ICAM1ITGALCA1CA2
Hydrochloric Acid SCHEMBL27702031 0.79 ITGB2 (0.60) ITGB2ICAM1ITGALCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4820691-A HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1989-04-11 US disclosed
EP-0296581-A2 Amino acid 1,2-diketo derivatives as renin inhibitors E.R. SQUIBB & SONS, INC. (US) 1988-12-28 EP disclosed