SCHEMBL7439181

SCHEMBL7439181

COc1ccc(C2CC(=O)N(O)C2)cc1OC1CCCC1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 14/20 0.77
PDE4B Q07343 16/20 0.63
PDE4C Q08493 10/20 0.63
PDE4D Q08499 10/20 0.63
CYP3A4 P08684 2/20 0.61
VEGFA P15692 1/20 0.61
ALDH1A1 P00352 1/20 0.61
LMNA P02545 1/20 0.61
CYP1A2 P05177 1/20 0.61
MAPT P10636 1/20 0.61
CYP2C9 P11712 1/20 0.61
ALOX15 P16050 1/20 0.61
CREBBP Q92793 1/20 0.61
KDM4E B2RXH2 1/20 0.61
PDE5A O76074 1/20 0.61
TNF P01375 1/20 0.61
MAPK1 P28482 1/20 0.61
BLM P54132 1/20 0.61
PDE1A P54750 1/20 0.61
PDE1B Q01064 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6755741 0.87 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL16774566 0.85 PDE4A (0.72) PDE4APDE4BPDE4CPDE4D
SCHEMBL30930191 0.85 PDE4A (0.72) PDE4APDE4BPDE4CPDE4D
SCHEMBL3549032 0.85 PDE4A (0.75) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL13986131 0.84 PDE4A (0.74) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL3542660 0.84 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL13654775 0.84 PDE4A (0.73) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL5227988 0.84 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL3539891 0.84 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DCYP3A4
SCHEMBL7365947 0.83 PDE4A (0.74) PDE4APDE4BPDE4CPDE4DCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3227155-B2 2001-11-12 JP claimed
EP-0526535-B1 CYCLIC HYDROXAMIC ACIDS AND THEIR USE ORION YHTYMAE OY (FI) 1995-09-27 EP claimed
US-5356923-A 1-hydroxy-4(3-cyclopentyloxy-4-methoxyphenyl)-2-pyrrolidone and anti-hypertensive use thereof ORION-YHTYMA OY (FI) 1994-10-18 US claimed
EP-0526535-A1 CYCLIC HYDROXAMIC ACIDS AND THEIR USE. ORION YHTYMAE OY (FI) 1993-02-10 EP claimed
WO-1991016303-A1 CYCLIC HYDROXAMIC ACIDS AND THEIR USE Orion-Yhtymä Oy (FI) 1991-10-31 WO claimed
US-11286280-B2 Melanocortin-1 receptor-specific peptides for cytokine storm and inflammation therapy PALATIN TECHNOLOGIES, INC. (US) 2022-03-29 US disclosed
EP-0675886-A1 AMINOMETHYLENE SUBSTITUTED NON-AROMATIC HETEROCYCLES AND USE AS SUBSTANCE P ANTAGONISTS PFIZER INC. (US) 1995-10-11 EP disclosed
EP-0526535-B1 CYCLIC HYDROXAMIC ACIDS AND THEIR USE ORION YHTYMAE OY (FI) 1995-09-27 EP disclosed
US-5356923-A 1-hydroxy-4(3-cyclopentyloxy-4-methoxyphenyl)-2-pyrrolidone and anti-hypertensive use thereof ORION-YHTYMA OY (FI) 1994-10-18 US disclosed
US-5356923-A 1-hydroxy-4(3-cyclopentyloxy-4-methoxyphenyl)-2-pyrrolidone and anti-hypertensive use thereof ORION-YHTYMA OY (FI) 1994-10-18 US disclosed
EP-0526535-A1 CYCLIC HYDROXAMIC ACIDS AND THEIR USE. ORION YHTYMAE OY (FI) 1993-02-10 EP disclosed
WO-1991016303-A1 CYCLIC HYDROXAMIC ACIDS AND THEIR USE Orion-Yhtymä Oy (FI) 1991-10-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11286280-B2 Melanocortin-1 receptor-specific peptides for cytokine storm and inflammation therapy MC3R, MC1R, MC2R PDE4A 1771/4885PDE4B 2513/4885PDE4C 2075/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.