SCHEMBL7439436

SCHEMBL7439436

CC(C)[C@H](NC(=O)N(C)Cc1nc2ccccc2[nH]1)C(=O)NC(Cc1ccccc1)C(O)C(O)C(Cc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.55
CTSD P07339 4/20 0.51
PTPN1 P18031 1/20 0.49
KLK5 Q9Y337 1/20 0.46
PSEN1 P49768 3/20 0.45
PSEN2 P49810 3/20 0.45
APH1B Q8WW43 3/20 0.45
NCSTN Q92542 3/20 0.45
APH1A Q96BI3 3/20 0.45
PSENEN Q9NZ42 3/20 0.45
BACE1 P56817 2/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9235504 1.00 CA2 (0.55) CA2CTSDPTPN1KLK5PSEN1
SCHEMBL7333388 0.92 CA2 (0.64) CA2CTSDCYP1A2CYP3A4CYP2D6
SCHEMBL7333130 0.92 CA2 (0.64) CA2CTSDCYP1A2CYP3A4CYP2D6
SCHEMBL7333674 0.92 CA2 (0.64) CA2CTSDCYP1A2CYP3A4CYP2D6
SCHEMBL7310994 0.82 CA2 (0.67) CA2CTSDBACE1CYP1A2CYP3A4
SCHEMBL7439444 0.82 PTPN1 (0.45) CTSDPTPN1KLK5PSEN1PSEN2
SCHEMBL7331805 0.81 CA2 (0.83) CA2KLK5PSEN1PSEN2APH1B
SCHEMBL7332653 0.81 CA2 (0.83) CA2KLK5PSEN1PSEN2APH1B
SCHEMBL7340722 0.81 CA2 (0.83) CA2KLK5PSEN1PSEN2APH1B
SCHEMBL7425008 0.80 CA2 (0.59) CA2KLK5PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018866-A2 1,4-DIAMINO-2,3-DIHYDROXYBUTANES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-12-12 WO claimed
EP-0665215-A1 1,4-Diamino-2,3-dihydroxybutanes THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-08-02 EP disclosed
WO-1991018866-A2 1,4-DIAMINO-2,3-DIHYDROXYBUTANES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-12-12 WO disclosed