SCHEMBL7439732

SCHEMBL7439732

CCC(c1cccs1)c1c(O)cc(CC2(CC3CCCCO3)CC2)oc1=O

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.36
HPGD P15428 2/20 0.35
KDM4E B2RXH2 5/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
POLB P06746 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MAPT P10636 3/20 0.34
TSHR P16473 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
LMNA P02545 2/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
KMT2A Q03164 3/20 0.33
HTT P42858 2/20 0.33
MEN1 O00255 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7445249 0.98 HPGD (0.36) ALDH1A1HPGDKDM4EPOLBHSD17B10
SCHEMBL7450257 0.88 ALDH1A1 (0.36) ALDH1A1HPGDKDM4EOPRM1OPRD1
SCHEMBL7440655 0.86 ALDH1A1 (0.37) ALDH1A1HPGDKDM4EPOLBMAPT
SCHEMBL7435600 0.86 NQO1 (0.31)
SCHEMBL7446268 0.86 HPGD (0.36) ALDH1A1HPGDKDM4EPOLBHSD17B10
SCHEMBL7438652 0.86 FEN1 (0.33) ALDH1A1KMT2AMEN1
SCHEMBL7445490 0.85 ERCC5 (0.31)
SCHEMBL7448075 0.84 ALDH1A1 (0.35) ALDH1A1HPGDKDM4EPOLBMAPT
SCHEMBL7481812 0.83 NQO1 (0.34)
SCHEMBL7447160 0.82 MAPT (0.34) ALDH1A1HPGDHSD17B10MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed