SCHEMBL7447160

SCHEMBL7447160

CCC(c1cccs1)c1c(O)cc(CC2(Cc3ccco3)CC2)oc1=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.34
NPSR1 Q6W5P4 4/20 0.34
HTT P42858 2/20 0.33
ALDH1A1 P00352 5/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
NQO1 P15559 1/20 0.33
TSHR P16473 3/20 0.32
OGT O15294 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
GAA P10253 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
ALOX15 P16050 1/20 0.31
CYP2C19 P33261 1/20 0.31
HSD17B10 Q99714 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7481812 0.89 NQO1 (0.34) NQO1CYP2C9
SCHEMBL7435521 0.86 NQO1 (0.31) NQO1
SCHEMBL7443467 0.86 MAPT (0.33) MAPTALDH1A1LMNATP53MEN1
SCHEMBL7449294 0.85 NQO1 (0.32) NQO1
SCHEMBL7443227 0.84 LMNA (0.33) MAPTNPSR1HTTALDH1A1LMNA
SCHEMBL7445249 0.84 HPGD (0.36) MAPTNPSR1HTTALDH1A1LMNA
SCHEMBL7439732 0.82 ALDH1A1 (0.36) MAPTNPSR1HTTALDH1A1LMNA
SCHEMBL7435600 0.82 NQO1 (0.31) NQO1
SCHEMBL7445490 0.81 ERCC5 (0.31) NQO1
SCHEMBL7438652 0.80 FEN1 (0.33) ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
CN-1040321-C Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating HIV and other retroviruses UPJOHN CO (US) 1998-10-21 CN disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed