SCHEMBL7440880

SCHEMBL7440880

COc1ccc(-c2cccc(C(CC(C)C)C(=O)NCC#N)c2S(=O)(=O)N2CCN(CCO)CC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSK P43235 18/20 0.52
CTSS P25774 18/20 0.52
CTSL P07711 14/20 0.52
CTSB P07858 13/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7440883 0.81 CTSK (0.62) CTSKCTSSCTSLCTSB
SCHEMBL7399589 0.78 CTSK (0.53) CTSKCTSSCTSLCTSB
SCHEMBL4711952 0.77 CTSK (0.67) CTSKCTSSCTSLCTSB
SCHEMBL6247222 0.74 CTSK (0.55) CTSKCTSSCTSLCTSB
SCHEMBL4712579 0.72 CTSK (0.64) CTSKCTSSCTSLCTSB
SCHEMBL6219216 0.70 CTSK (0.58) CTSKCTSSCTSLCTSB
SCHEMBL4716242 0.69 CTSK (0.72) CTSKCTSSCTSLCTSB
SCHEMBL6247225 0.69 CTSK (0.65) CTSKCTSSCTSLCTSB
SCHEMBL4713554 0.69 CTSK (1.00) CTSKCTSSCTSLCTSB
SCHEMBL4713043 0.68 CTSK (0.81) CTSKCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001049288-A9 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2001-10-25 WO disclosed