SCHEMBL7441256

SCHEMBL7441256

CCNC(=O)Nc1cccc(-c2c3nn(-c4ccc(Cl)cc4)c(=O)c-3c[nH]c2C)c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PSD A5PKW4 2/20 0.44
CNR1 P21554 13/20 0.41
CDK8 P49336 1/20 0.41
MAPT P10636 1/20 0.38
CNR2 P34972 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA7 P43166 1/20 0.38
FGFR3 P22607 1/20 0.38
KDR P35968 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7439496 0.82 PTGS2 (0.45)
SCHEMBL2650293 0.82 PTDSS1 (0.38) CNR1MAPT
SCHEMBL2649310 0.81 CSNK2A1 (0.42) PSDMAPT
SCHEMBL2649769 0.81 DHODH (0.44) CNR1MAPT
SCHEMBL2648853 0.79 GAA (0.39) PSDMAPTCA1CA2KDR
SCHEMBL2649751 0.79 KIT (0.40) PSDMAPTKDR
SCHEMBL2650770 0.78 GAA (0.47) MAPTCA1CA2KDR
SCHEMBL2651418 0.78 ABCB1 (0.43) PSDMAPTKDR
Hydrochloric Acid SCHEMBL2662150 0.77 GAA (0.46) MAPTCA1CA2KDR
SCHEMBL2649448 0.77 DHODH (0.40) MAPTKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6333336-B1 GAMMA-AMINOBUTYRIC ACID RECEPTORS AS ANTICONVULSANTS FORMING THE COMPOUND BY AMIDATION MERCK SHARP & DOHME LTD. (GB) 2001-12-25 US claimed
US-6333336-B1 GAMMA-AMINOBUTYRIC ACID RECEPTORS AS ANTICONVULSANTS FORMING THE COMPOUND BY AMIDATION MERCK SHARP & DOHME LTD. (GB) 2001-12-25 US disclosed