SCHEMBL7443597

SCHEMBL7443597

CCC(c1cccs1)c1c(O)cc(C(Cc2ccc(Cl)cc2)CC2CC2)oc1=O

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.34
ALDH1A1 P00352 1/20 0.34
NQO1 P15559 1/20 0.33
MME P08473 1/20 0.32
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
MEN1 O00255 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
NPY5R Q15761 1/20 0.30
TP53 P04637 1/20 0.30
PPARG P37231 1/20 0.30
PPARA Q07869 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7451071 0.93 NQO1 (0.34) NQO1CYP2C9
SCHEMBL7440329 0.92 NQO1 (0.33) NQO1NPY5RCYP2C9
SCHEMBL7437094 0.92 NQO1 (0.33) ALDH1A1NQO1MEN1KMT2ANPY5R
SCHEMBL7440406 0.91 NQO1 (0.33) NQO1MEN1KMT2ATP53CYP2C9
SCHEMBL7439255 0.90 MAPT (0.37) MAPTALDH1A1NQO1MMEKDM4E
SCHEMBL7443735 0.90 TP53 (0.35) MAPTALDH1A1NQO1POLBMEN1
SCHEMBL7440164 0.90 CNR1 (0.34) NQO1PPARGPPARA
SCHEMBL9281720 0.90 CNR1 (0.34) NQO1PPARGPPARA
SCHEMBL7450255 0.87 NQO1 (0.33) MAPTNQO1NPY5RTP53
SCHEMBL7437064 0.86 MAPT (0.36) MAPTALDH1A1MEN1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed