SCHEMBL7444044

SCHEMBL7444044

CC(CCNC(=O)c1cccc(-c2csc(NC(=N)N)n2)c1)CC(=O)NCC#N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 3/20 0.41
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
STAT3 P40763 1/20 0.41
MAPT P10636 6/20 0.40
ALDH1A1 P00352 4/20 0.40
THRB P10828 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
GAA P10253 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PRKD1 Q15139 1/20 0.39
CSNK2A2 P19784 1/20 0.39
CSNK2B P67870 1/20 0.39
CSNK2A1 P68400 1/20 0.39
CSNK2A3 Q8NEV1 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6181733 0.91 KMT2A (0.47) ABL1MEN1KMT2ASTAT3MAPT
SCHEMBL7455830 0.82 KMT2A (0.44) ABL1MEN1KMT2ASTAT3MAPT
SCHEMBL6184390 0.81 CTSL (0.59)
SCHEMBL6183646 0.79 PARP1 (0.52) MEN1KMT2ASTAT3MAPTALDH1A1
SCHEMBL7452212 0.78 KMT2A (0.44) MEN1KMT2AMAPTALDH1A1NPC1
SCHEMBL6183920 0.77 NPC1 (0.45) MEN1KMT2AMAPTALDH1A1NPC1
SCHEMBL7450325 0.77 ALDH1A1 (0.47) MEN1KMT2AMAPTALDH1A1NPC1
SCHEMBL11091588 0.76 MAPT (0.55) ABL1MEN1KMT2AMAPTALDH1A1
SCHEMBL7453120 0.76 NAMPT (0.41) NPC1RAB9AHTTSMN1; SMN2
SCHEMBL7452860 0.75 KDM4E (0.60) MEN1KMT2AMAPTALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161415-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-12 EP disclosed
WO-2000055126-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed