SCHEMBL7444732

SCHEMBL7444732

COc1[c]noc1-c1cccs1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 10/20 0.40
RAB9A P51151 10/20 0.40
KDM4E B2RXH2 5/20 0.40
PKM P14618 2/20 0.40
MAPT P10636 2/20 0.40
SMN1; SMN2 Q16637 7/20 0.40
ALDH1A1 P00352 6/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
RPS6KB2 Q9UBS0 2/20 0.40
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
MAPK1 P28482 4/20 0.38
HSD17B10 Q99714 4/20 0.38
TP53 P04637 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
CASP3 P42574 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4767260 0.73 PTGS1 (0.37) NPC1RAB9AMAPTSMN1; SMN2ALDH1A1
SCHEMBL4150903 0.72 CYP2C9 (0.40) NPC1RAB9AKDM4EMAPTSMN1; SMN2
SCHEMBL7451095 0.71 SMPD3 (0.40) ADORA2AADORA1
SCHEMBL7453983 0.70 RPS6KB2 (0.41) NPC1RAB9AKDM4EPKMMAPT
SCHEMBL7112445 0.69 CLK4 (0.36) NPC1RAB9AKDM4EPKMMAPT
SCHEMBL9769080 0.69 ALDH1A1 (0.50) NPC1RAB9AKDM4EPKMMAPT
SCHEMBL7105969 0.68 NPC1 (0.40) NPC1RAB9AKDM4EPKMMAPT
SCHEMBL3220235 0.67 RAB9A (0.39) NPC1RAB9AKDM4EPKMMAPT
SCHEMBL7455270 0.64 KDM4E (0.40) NPC1RAB9AKDM4EPKMMAPT
SCHEMBL19127576 0.63 ERN1 (0.40) NPC1RAB9AKDM4EPKMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1104403-A1 HYDROXY PIPECOLATE HYDROXAMIC ACID DERIVATIVES AS MMP INHIBITORS Pfizer Products Inc. (US) 2001-06-06 EP disclosed
WO-2000009485-A1 HYDROXY PIPECOLATE HYDROXAMIC ACID DERIVATIVES AS MMP INHIBITORS PFIZER PRODUCTS INC. (US) 2000-02-24 WO disclosed