SCHEMBL7445219

SCHEMBL7445219

CCOC(=O)CCCN(c1c(C)cccc1C(=O)NO)S(=O)(=O)c1ccc(OC)cc1

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 18/20 0.66
MMP1 P03956 17/20 0.66
MMP9 P14780 17/20 0.66
ADAM17 P78536 10/20 0.65
BMP1 P13497 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7446698 0.97 MMP13 (0.65) MMP13MMP1MMP9ADAM17
SCHEMBL27510654 0.86 MMP13 (0.70) MMP13MMP1MMP9ADAM17BMP1
SCHEMBL27510267 0.86 MMP13 (0.70) MMP13MMP1MMP9ADAM17BMP1
SCHEMBL7313705 0.85 MMP13 (0.74) MMP13MMP1MMP9ADAM17
SCHEMBL7323902 0.80 MMP13 (1.00) MMP13MMP1MMP9ADAM17
SCHEMBL7509702 0.79 MMP13 (0.76) MMP13MMP1MMP9ADAM17
SCHEMBL7320844 0.79 MMP13 (1.00) MMP13MMP1MMP9ADAM17
SCHEMBL7322084 0.79 MMP13 (0.82) MMP13MMP1MMP9ADAM17
SCHEMBL7443729 0.78 MMP13 (1.00) MMP13MMP1MMP9ADAM17
SCHEMBL7004444 0.78 BMP1 (0.71) BMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0938471-B1 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS AMERICAN CYANAMID CO (US) 2001-12-12 EP claimed
EP-0938471-A1 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS American Cyanamid Company (US) 1999-09-01 EP claimed
WO-1998016503-A2 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS AMERICAN CYANAMID COMPANY (US) 1998-04-23 WO claimed
EP-0938471-B1 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS AMERICAN CYANAMID CO (US) 2001-12-12 EP disclosed
EP-0938471-A1 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS American Cyanamid Company (US) 1999-09-01 EP disclosed
WO-1998016503-A2 THE PREPARATION AND USE OF ORTHO-SULFONAMIDO ARYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASE AND TACE INHIBITORS AMERICAN CYANAMID COMPANY (US) 1998-04-23 WO disclosed