SCHEMBL7445322

SCHEMBL7445322

COc1cc2c(C)nc(O)c(NC(C)=O)c2cc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
TSHR P16473 1/20 0.47
HSD17B10 Q99714 4/20 0.45
KDM4E B2RXH2 2/20 0.45
MAPT P10636 2/20 0.45
SAE1 Q9UBE0 1/20 0.45
UBA2 Q9UBT2 1/20 0.45
ATM Q13315 1/20 0.41
GAA P10253 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
POLB P06746 1/20 0.41
EGFR P00533 1/20 0.41
KDR P35968 1/20 0.41
CYP1A2 P05177 1/20 0.41
ADORA3 P0DMS8 2/20 0.40
LMNA P02545 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAPK1 P28482 3/20 0.39
CASP3 P42574 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL9830179 0.99 ALDH1A1 (0.46) ALDH1A1TSHRHSD17B10KDM4EMAPT
Water SCHEMBL9830187 0.99 ALDH1A1 (0.46) ALDH1A1TSHRHSD17B10KDM4EMAPT
SCHEMBL9831668 0.87 KMT2A (0.40) ALDH1A1TSHRKDM4EMAPTGAA
SCHEMBL9832514 0.85 KDM4E (0.42) ALDH1A1TSHRHSD17B10KDM4EMAPT
SCHEMBL7413138 0.82 ALDH1A1 (0.41) ALDH1A1TSHRHSD17B10KDM4EMAPT
SCHEMBL9832403 0.79 EGFR (0.49) ALDH1A1TSHRHSD17B10KDM4EMAPT
SCHEMBL9831559 0.79 KDR (0.49) ALDH1A1TSHRHSD17B10KDM4EMAPT
SCHEMBL9830353 0.79 GAA (0.40) ALDH1A1KDM4EMAPTGAAMEN1
SCHEMBL9831858 0.79 CA12 (0.50) ALDH1A1HSD17B10KDM4EMAPTGAA
Water SCHEMBL10786992 0.78 KDR (0.48) ALDH1A1TSHRHSD17B10KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4880817-A O-functionalized derivatives of substituted isoquinolin-3-ols having cardiotonic and/or phosphodiesterase fraction III inhibiting properties and/or renal vasodilating properties ORTHO PHARMACEUTICAL CORPORATION (US) 1989-11-14 US disclosed