SCHEMBL7413138

SCHEMBL7413138

COc1cc2c(C)nc(N(C)C)c(NC(C)=O)c2cc1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 3/20 0.39
KDM4E B2RXH2 3/20 0.39
MAPT P10636 2/20 0.39
SAE1 Q9UBE0 1/20 0.39
UBA2 Q9UBT2 1/20 0.39
ATM Q13315 1/20 0.39
EGFR P00533 1/20 0.39
KDR P35968 1/20 0.39
CYP1A2 P05177 2/20 0.38
ADORA3 P0DMS8 3/20 0.38
LMNA P02545 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
SENP7 Q9BQF6 3/20 0.37
SENP6 Q9GZR1 3/20 0.37
CASP3 P42574 2/20 0.37
SENP8 Q96LD8 2/20 0.37
MAPK1 P28482 2/20 0.37
GAA P10253 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7445322 0.82 ALDH1A1 (0.47) ALDH1A1TSHRHSD17B10KDM4EMAPT
Water SCHEMBL9830187 0.81 ALDH1A1 (0.46) ALDH1A1TSHRHSD17B10KDM4EMAPT
Water SCHEMBL9830179 0.81 ALDH1A1 (0.46) ALDH1A1TSHRHSD17B10KDM4EMAPT
SCHEMBL7409180 0.72 MAPT (0.43) ALDH1A1HSD17B10KDM4EMAPTLMNA
SCHEMBL7409625 0.72 KMT2A (0.45) ALDH1A1HSD17B10KDM4EMAPTEGFR
SCHEMBL9831668 0.69 KMT2A (0.40) ALDH1A1TSHRKDM4EMAPTLMNA
SCHEMBL9832514 0.68 KDM4E (0.42) ALDH1A1TSHRHSD17B10KDM4EMAPT
SCHEMBL10683659 0.66 HSD17B10 (0.47) ALDH1A1TSHRHSD17B10KDM4EMAPT
SCHEMBL12325390 0.65 CYP3A4 (0.46) ALDH1A1TSHRKDM4EMAPTLMNA
SCHEMBL16582707 0.65 SENP7 (0.44) ALDH1A1HSD17B10KDM4EMAPTSAE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4843077-A Isoquinoline derivatives having renal vasodilating properties and/or cardiotonic properties and/or phosphodiesterase inhibiting properties ORTHO PHARMACEUTICAL CORPORATION (US) 1989-06-27 US disclosed