SCHEMBL7445482

SCHEMBL7445482

CCC(NS(=O)(=O)c1cc(Cl)cc(Cl)c1)C(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MME P08473 8/20 0.58
ACE P12821 6/20 0.58
CPA1 P15085 3/20 0.58
ACE2 Q9BYF1 3/20 0.58
CA2 P00918 1/20 0.51
ITGB1 P05556 1/20 0.49
ITGA4 P13612 1/20 0.49
ADAMTS5 Q9UNA0 1/20 0.46
MMP2 P08253 1/20 0.46
PIN1 Q13526 2/20 0.44
PTPN1 P18031 1/20 0.44
MMP9 P14780 1/20 0.44
MMP8 P22894 1/20 0.44
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
POLB P06746 1/20 0.43
F2 P00734 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7444227 0.80 ITGB1 (0.55) CA2ITGB1ITGA4ADAMTS5MMP2
SCHEMBL7447944 0.78 MME (0.52) MMEACECPA1ACE2CA2
SCHEMBL7442952 0.78 ITGB1 (0.53) ACECA2ITGB1ITGA4ADAMTS5
SCHEMBL7360349 0.77 MMP2 (0.72) ITGB1ITGA4ADAMTS5MMP2MMP9
SCHEMBL7381453 0.77 MMP2 (0.72) ITGB1ITGA4ADAMTS5MMP2MMP9
SCHEMBL7448892 0.76 MMP2 (0.53) ACECA2ITGB1ITGA4ADAMTS5
SCHEMBL15342313 0.76 MME (0.60) MMEACECPA1ACE2CA2
SCHEMBL29386041 0.76 MME (0.60) MMEACECPA1ACE2CA2
SCHEMBL7298796 0.76 MMP2 (0.70) ADAMTS5MMP2MMP9POLBF2
SCHEMBL31296488 0.75 MME (0.71) MMEACECPA1ACE2CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0977743-A1 PROTEASE INHIBITORS Smithkline Beecham (US) 2000-02-09 EP disclosed
WO-1998049152-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1998-11-05 WO disclosed