SCHEMBL7446445

SCHEMBL7446445

CCOC(=O)CNC(C)(C(=O)N1CCCC1)c1ccc2[nH]c(CNc3ccc(C#N)cc3)nc2c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.38
ALDH1A1 P00352 2/20 0.38
RAB9A P51151 2/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
F2 P00734 1/20 0.35
F10 P00742 1/20 0.35
MLLT1 Q03111 1/20 0.34
P2RY12 Q9H244 1/20 0.34
DGAT2 Q96PD7 1/20 0.33
PIP4K2A P48426 1/20 0.33
TGFBR1 P36897 2/20 0.32
IDH1 O75874 2/20 0.31
CHEK1 O14757 1/20 0.31
POLB P06746 1/20 0.31
HTR1A P08908 2/20 0.31
USP14 P54578 1/20 0.31
HRH2 P25021 1/20 0.31
HRH1 P35367 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7454489 1.00 NPC1 (0.38) NPC1ALDH1A1RAB9ALMNAMAPT
SCHEMBL7447136 0.93 ALDH1A1 (0.37) NPC1ALDH1A1RAB9ALMNAMAPT
SCHEMBL7447505 0.92 NPC1 (0.36) NPC1ALDH1A1RAB9ALMNAMAPT
SCHEMBL7442305 0.88 F2 (0.48) NPC1ALDH1A1RAB9ALMNAMAPT
Hydrochloric Acid SCHEMBL7449029 0.87 F2 (0.47) NPC1ALDH1A1RAB9ALMNAMAPT
Hydrochloric Acid SCHEMBL7418107 0.87 F2 (0.47) NPC1ALDH1A1RAB9ALMNAMAPT
SCHEMBL7453448 0.87 RAB9A (0.41) NPC1ALDH1A1RAB9ALMNAMAPT
SCHEMBL7449129 0.86 RAB9A (0.40) NPC1ALDH1A1RAB9ALMNAMAPT
SCHEMBL7421109 0.85 NPC1 (0.37) NPC1ALDH1A1RAB9ALMNAMAPT
SCHEMBL7442673 0.85 MLLT1 (0.34) NPC1ALDH1A1RAB9ALMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095025-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-05-02 EP disclosed
WO-2000001704-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-01-13 WO disclosed