SCHEMBL7446807

SCHEMBL7446807

Cc1cc(C)c(S(=O)(=O)NC(CNC(=O)c2ccc(-c3cccc(N)c3)s2)C(=O)OC(C)(C)C)c(C)c1

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 15/20 0.62
ITGB3 P05106 12/20 0.62
ITGA2B P08514 10/20 0.62
ITGB1 P05556 7/20 0.62
ITGA5 P08648 7/20 0.62
ITGB5 P18084 7/20 0.62
HPGDS O60760 2/20 0.43
ESR1 P03372 2/20 0.40
ESRRG P62508 2/20 0.40
ESR2 Q92731 2/20 0.40
ACKR3 P25106 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7448307 0.87 ITGB3 (0.58) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7455544 0.83 ITGAV (0.51) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7976674 0.83 ITGAV (0.51) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7455550 0.83 ITGAV (0.51) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7447358 0.82 ITGAV (0.56) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7452852 0.81 ITGB3 (0.57) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL6016242 0.81 ITGAV (0.53) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7455915 0.78 ITGB3 (0.53) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7962800 0.78 ITGB3 (0.53) ITGAVITGB3ITGA2BITGB1ITGA5
SCHEMBL7448645 0.78 ITGB3 (0.59) ITGAVITGB3ITGA2BITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187825-A1 THIOPHENE INTEGRIN INHIBITORS Shire Biochem Inc. (CA) 2002-03-20 EP disclosed
WO-2000075129-A1 THIOPHENE INTEGRIN INHIBITORS SHIRE BIOCHEM INC. (CA) 2000-12-14 WO disclosed