SCHEMBL744779

SCHEMBL744779

O=C(O)[C@@H](Br)c1ccccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.48
SLC6A3 Q01959 2/20 0.48
SLC6A2 P23975 1/20 0.48
SLC6A4 P31645 1/20 0.48
ALDH1A1 P00352 3/20 0.47
CYP1A2 P05177 2/20 0.47
KDM4E B2RXH2 3/20 0.47
NPSR1 Q6W5P4 1/20 0.46
LMNA P02545 3/20 0.45
NAPRT Q6XQN6 1/20 0.45
P4HTM Q9NXG6 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
CYP3A4 P08684 3/20 0.45
PTPRA P18433 1/20 0.44
CES2 O00748 2/20 0.42
CES1 P23141 2/20 0.42
TSHR P16473 3/20 0.41
ABCB11 O95342 1/20 0.41
ESR1 P03372 1/20 0.41
ADRA2A P08913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3638184 1.00 GSK3B (0.48) GSK3BSLC6A3SLC6A2SLC6A4ALDH1A1
SCHEMBL6510710 0.83 CYP1A2 (0.53) GSK3BSLC6A3SLC6A2SLC6A4ALDH1A1
Bromide SCHEMBL6278361 0.82 CYP1A2 (0.51) GSK3BSLC6A3SLC6A2SLC6A4ALDH1A1
SCHEMBL3767996 0.79 SLC6A3 (0.52) GSK3BSLC6A3SLC6A2SLC6A4ALDH1A1
SCHEMBL7719801 0.79 ALDH1A1 (0.59) GSK3BSLC6A3SLC6A2SLC6A4ALDH1A1
SCHEMBL11146589 0.78 CYP2C19 (0.55) GSK3BSLC6A3SLC6A2SLC6A4ALDH1A1
SCHEMBL75590 0.78 KMT2A (0.47) GSK3BSLC6A3SLC6A2SLC6A4ALDH1A1
SCHEMBL10170706 0.78 KDM4E (0.53) GSK3BSLC6A3SLC6A2SLC6A4ALDH1A1
SCHEMBL6638556 0.78 SLC6A3 (0.50) GSK3BSLC6A3SLC6A2SLC6A4ALDH1A1
SCHEMBL1685422 0.78 KDM4E (0.53) GSK3BSLC6A3SLC6A2SLC6A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430018-A2 BENZOXAZOLONE DERIVATIVES AS ALDOSTERONE SYMTHASE INHIBITORS Novartis AG (CH) 2012-03-21 EP disclosed
WO-2010130773-A2 BENZOXAZOLONE DERIVATIVES AS ALDOSTERONE SYMTHASE INHIBITORS NOVARTIS AG (CH) 2010-11-18 WO disclosed