SCHEMBL7447953

SCHEMBL7447953

CC(C)CCN(C(=O)c1ccc(NC(=O)O)cc1)C(=O)N(C)C#N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.43
NPC1 O15118 2/20 0.37
GAA P10253 1/20 0.37
PKM P14618 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ALDH1A1 P00352 2/20 0.36
ADRB2 P07550 1/20 0.36
HTT P42858 1/20 0.36
CTSL P07711 2/20 0.35
CTSB P07858 2/20 0.35
CTSS P25774 2/20 0.35
CTSK P43235 2/20 0.35
HPGD P15428 2/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7452320 0.83 F2 (0.35) NAMPTNPC1HSD17B10ALDH1A1CTSS
SCHEMBL7447948 0.82 NAMPT (0.40) NAMPTNPC1PKMMAPK1HSD17B10
SCHEMBL6257637 0.81 NAMPT (0.33) NAMPTNPC1ALDH1A1CTSBLPAR1
SCHEMBL7486324 0.79 FAAH (0.53) NAMPTNPC1MAPK1RAB9A
SCHEMBL6251138 0.78 GRIK1 (0.38) ADRB2LPAR1LPAR5
SCHEMBL6182144 0.78 NAMPT (0.46) NAMPTNPC1GAAALDH1A1MEN1
SCHEMBL6183130 0.77 GAA (0.49) NAMPTGAAMAPK1HSD17B10ALDH1A1
SCHEMBL6183489 0.77 NAMPT (0.46) NAMPTNPC1ALDH1A1MEN1KMT2A
SCHEMBL6255637 0.76 LPAR1 (0.31) ALDH1A1CTSBMEN1KMT2ALPAR1
SCHEMBL6252192 0.75 SRD5A2 (0.47) CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2002539192-A 2002-11-19 JP claimed
EP-1161415-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-12 EP claimed
WO-2000055126-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO claimed