SCHEMBL7447948

SCHEMBL7447948

CC(C)CCN(C(=O)NCC#N)C(=O)c1ccc(NC(=O)O)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.40
CTSL P07711 6/20 0.37
CTSB P07858 4/20 0.37
CTSS P25774 5/20 0.36
CTSK P43235 1/20 0.36
PKM P14618 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ALDH1A1 P00352 1/20 0.35
ADRB2 P07550 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
THRB P10828 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6876209 0.87 CASR (0.42) CTSLCTSBCTSSCTSKHSD17B10
SCHEMBL7447953 0.82 NAMPT (0.43) NAMPTCTSLCTSBCTSSCTSK
SCHEMBL6182151 0.78 NAMPT (0.44) NAMPTCTSSALDH1A1LMNATP53
SCHEMBL6183132 0.77 GAA (0.48) NAMPTMAPK1HSD17B10ALDH1A1LMNA
SCHEMBL6183497 0.77 CNR2 (0.44) NAMPTALDH1A1NPC1RAB9ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL6182101 0.76 PRKAB2 (0.49) NAMPTMAPK1
SCHEMBL6183364 0.76 CTSB (0.35) CTSLCTSBCTSSCTSKNPC1
SCHEMBL6183242 0.75 CTSK (0.37) CTSLCTSBCTSSCTSK
SCHEMBL5521755 0.73 PRMT5 (0.42) CTSLCTSBCTSSCTSKHDAC1
SCHEMBL6184516 0.71 KDM4E (0.44) NAMPTALDH1A1LMNANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2002539192-A 2002-11-19 JP claimed
EP-1161415-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-12 EP claimed
WO-2000055126-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO claimed