SCHEMBL7448733

SCHEMBL7448733

O=C(NCc1ccccc1)c1ccc2n[c]sc2c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.62
ADORA3 P0DMS8 1/20 0.62
ADORA2A P29274 1/20 0.62
ADORA2B P29275 1/20 0.62
ADORA1 P30542 1/20 0.62
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
PLAU P00749 1/20 0.56
HDAC1 Q13547 2/20 0.54
HPGD P15428 3/20 0.53
ALDH1A1 P00352 2/20 0.53
KDM4E B2RXH2 1/20 0.53
MEN1 O00255 1/20 0.53
POLB P06746 1/20 0.53
MAPT P10636 1/20 0.53
THRB P10828 1/20 0.53
PTPN7 P35236 1/20 0.53
RECQL P46063 1/20 0.53
BLM P54132 1/20 0.53
KMT2A Q03164 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7448662 0.84 HPGD (0.53) CYP2D6HPGDALDH1A1MEN1POLB
SCHEMBL7452674 0.81 RAB9A (0.65) PLAUHDAC1HPGDALDH1A1KDM4E
SCHEMBL7456577 0.79 KDM4E (0.64) CYP2D6ADORA3ADORA2AADORA2BADORA1
SCHEMBL27306157 0.78 CYP2D6 (0.76) CYP2D6ADORA3ADORA2AADORA2BADORA1
SCHEMBL13491477 0.77 CYP2D6 (0.74) CYP2D6ADORA3ADORA2AADORA2BADORA1
SCHEMBL21177838 0.77 CYP2D6 (1.00) CYP2D6CYP2C9CYP2C19PLAUHDAC1
SCHEMBL7506844 0.76 NPC1 (0.44) CYP2D6CYP2C9CYP2C19PLAUHPGD
SCHEMBL7481830 0.75 ADORA3 (0.57) CYP2D6ADORA3ADORA2AADORA2BADORA1
SCHEMBL7451636 0.75 MEN1 (0.51) HPGDALDH1A1KDM4EMEN1POLB
SCHEMBL13491634 0.75 CYP2D6 (0.71) CYP2D6ADORA3ADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001027096-A9 AMINOMETHYL-(HETERO)ARYL DERIVATIVES AND THEIR USE AS TRYPTASE INHIBITORS PROTHERICS MOLECULAR DESIGN LT (GB) 2001-07-12 WO disclosed