SCHEMBL7448759

SCHEMBL7448759

COC(=O)C[C@H]1C(=O)N(CC(=O)OC)CCN1C(=O)CCC(=O)N1CCN(c2ccncc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 8/20 0.45
ITGA2B P08514 8/20 0.45
MMP2 P08253 1/20 0.41
CYP2D6 P10635 2/20 0.40
TSHR P16473 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CHRM1 P11229 2/20 0.38
FAP Q12884 1/20 0.38
HIF1A Q16665 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7448765 1.00 ITGB3 (0.45) ITGB3ITGA2BMMP2CYP2D6TSHR
SCHEMBL7368990 0.94 ITGB3 (0.51) ITGB3ITGA2BMMP2
SCHEMBL7368980 0.94 ITGB3 (0.51) ITGB3ITGA2BMMP2
SCHEMBL7366256 0.86 KDM4E (0.44) ITGB3ITGA2BMMP2TSHRCYP3A4
SCHEMBL7366261 0.86 KDM4E (0.44) ITGB3ITGA2BMMP2TSHRCYP3A4
SCHEMBL7368983 0.85 CYP2D6 (0.41) ITGB3ITGA2BMMP2CYP2D6TSHR
SCHEMBL7368598 0.84 KDM4E (0.52) TSHRCYP3A4CYP2C9ALDH1A1HSD17B10
SCHEMBL7368594 0.84 KDM4E (0.52) TSHRCYP3A4CYP2C9ALDH1A1HSD17B10
SCHEMBL7370702 0.82 ITGB3 (0.46) ITGB3ITGA2BCYP2D6TSHRCYP3A4
SCHEMBL7935145 0.82 ITGB3 (0.46) ITGB3ITGA2BCYP2D6TSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242600-B1 ANTIISCHEMIC AGENTS, ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-06-05 US disclosed
EP-0970071-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 2000-01-12 EP disclosed
WO-1998039324-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-11 WO disclosed