SCHEMBL7448764

SCHEMBL7448764

O=C(O)CC1NC(=O)C(Cc2ccc3ccccc3c2)NC1=O

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 7/20 0.47
CYP1A2 P05177 1/20 0.47
TACR2 P21452 1/20 0.43
OPRK1 P41145 3/20 0.42
OPRM1 P35372 1/20 0.42
OPRD1 P41143 1/20 0.42
SLC13A5 Q86YT5 1/20 0.41
NR1H4 Q96RI1 1/20 0.41
MMP13 P45452 1/20 0.41
AKR1B1 P15121 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
SIRT1 Q96EB6 1/20 0.40
SIRT3 Q9NTG7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1226564 0.83 ITGB3 (0.48)
SCHEMBL9021101 0.83 ITGB3 (0.48)
SCHEMBL3956081 0.83 ITGB3 (0.48)
SCHEMBL7456041 0.79 CXCR4 (0.43) CXCR4CYP1A2SIRT2SIRT1SIRT3
SCHEMBL8079346 0.78 CXCR4 (0.60) CXCR4CYP1A2TACR2OPRM1MMP13
SCHEMBL7456058 0.77 MMP1 (0.61) CXCR4CYP1A2
SCHEMBL10327213 0.75 CXCR4 (0.47) CXCR4
SCHEMBL7448481 0.75 CXCR4 (0.43) CXCR4CYP1A2TACR2OPRM1MMP13
SCHEMBL17676894 0.75 CXCR4 (0.47) CXCR4
SCHEMBL10327192 0.75 CXCR4 (0.47) CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001027096-A9 AMINOMETHYL-(HETERO)ARYL DERIVATIVES AND THEIR USE AS TRYPTASE INHIBITORS PROTHERICS MOLECULAR DESIGN LT (GB) 2001-07-12 WO disclosed