SCHEMBL7449167

SCHEMBL7449167

Cc1ccc2c(c1)[N]C=N2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.36
CYP2A6 P11509 3/20 0.36
GAA P10253 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HTT P42858 1/20 0.33
TP53 P04637 3/20 0.32
MAPT P10636 3/20 0.32
ALOX15 P16050 2/20 0.32
KMT2A Q03164 2/20 0.32
NQO2 P16083 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
ALOX12 P18054 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TDP1 Q9NUW8 6/20 0.32
CYP3A4 P08684 1/20 0.32
THRB P10828 1/20 0.32
TRPA1 O75762 1/20 0.32
ACHE P22303 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6365886 0.72
SCHEMBL207132 0.71 CA3 (0.31) CYP1A2CYP2A6ALDH1A1
SCHEMBL4273814 0.71 CA12 (0.40) CYP1A2CYP2A6SMN1; SMN2MAPTKMT2A
SCHEMBL24891183 0.70 CYP1A2 (0.35) CYP1A2CYP2A6GAASMN1; SMN2HTT
SCHEMBL208894 0.62 CA3 (0.31) CYP1A2CYP2A6ALDH1A1
SCHEMBL22028030 0.62 CYP3A4 (0.38) HTTMAPTALOX15KMT2AMEN1
SCHEMBL407343 0.62 NQO2 (0.37) CYP1A2CYP2A6GAASMN1; SMN2HTT
SCHEMBL10469300 0.62 NQO2 (0.37) CYP1A2CYP2A6GAASMN1; SMN2HTT
SCHEMBL21797549 0.62
SCHEMBL23537533 0.62 CYP1A2 (0.41) CYP1A2CYP2A6SMN1; SMN2TP53ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0744948-A4 PROTEASE INHIBITORS LILLY CO ELI (US) 1997-06-11 EP disclosed
US-5624934-A PREVENTING HIV INFECTION ELI LILLY AND COMPANY (US) 1997-04-29 US disclosed
EP-0744948-A1 PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 1996-12-04 EP disclosed
US-5480887-A FOR HIV, THIENO(3,2-C)PYRIDINE-(6S)-CARBOXAMIDES ELI LILLY AND COMPANY (US) 1996-01-02 US disclosed
WO-1995020962-A1 PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 1995-08-10 WO disclosed
US-4434174-A Treating cardiovascular diseases with N-(3-phenoxy-2-hydroxypropyl)benzimidazole-1-alkanamines BERLEX LABORATORIES, INC. (US) 1984-02-28 US disclosed
US-4363808-A N-(3-Phenoxy-2-hydroxypropyl)benzimidazole-1-alkanamines BERLEX LABORATORIES, INC. (US) 1982-12-14 US disclosed
EP-0034116-A2 N-(3-phenoxy-2-hydroxypropyl)benzimidazole-1-alkanamines BERLEX LABORATORIES, INC. (US) 1981-08-19 EP disclosed