SCHEMBL7449231

SCHEMBL7449231

O=C(Cc1ccccc1)Nc1cccs1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.60
KMT2A Q03164 4/20 0.60
MEN1 O00255 3/20 0.60
EPHX2 P34913 1/20 0.58
HPGD P15428 3/20 0.56
RAB9A P51151 2/20 0.56
MAPT P10636 2/20 0.56
ALDH1A1 P00352 2/20 0.56
NPC1 O15118 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
HSD17B10 Q99714 1/20 0.56
MAPK8 P45983 4/20 0.55
LMNA P02545 1/20 0.55
TP53 P04637 1/20 0.55
MAPK10 P53779 3/20 0.54
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11632220 0.82 ROCK1 (0.55) KDM4EKMT2AMEN1RAB9AMAPT
SCHEMBL9382436 0.77 GAA (0.51) KDM4EKMT2AMEN1HPGDRAB9A
SCHEMBL8853392 0.77 CASP3 (0.57) KDM4EKMT2AMEN1HPGDRAB9A
SCHEMBL3422728 0.77 GAA (0.55) KDM4EKMT2AMEN1HPGDRAB9A
SCHEMBL7351218 0.76 POLB (0.57) KMT2AMEN1RAB9AMAPTALDH1A1
SCHEMBL17384015 0.75 MEN1 (0.61) KDM4EKMT2AMEN1MAPTALDH1A1
Benzene SCHEMBL29129490 0.75 GAA (0.58) KDM4EKMT2AMEN1HPGDRAB9A
SCHEMBL418428 0.75
Hydrochloric Acid SCHEMBL28317066 0.75 GAA (0.54) KDM4EKMT2AMEN1HPGDRAB9A
Acetic Acid SCHEMBL10585627 0.75 GAA (0.49) KDM4EKMT2AMEN1HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0977743-A1 PROTEASE INHIBITORS Smithkline Beecham (US) 2000-02-09 EP disclosed
WO-1998049152-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1998-11-05 WO disclosed