SCHEMBL7449274

SCHEMBL7449274

Cc1c(CO)oc2cc(C#N)ccc12

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 2/20 0.44
MAOB P27338 10/20 0.44
IDO1 P14902 2/20 0.40
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
KLK7 P49862 1/20 0.38
ATM Q13315 1/20 0.38
ACHE P22303 1/20 0.38
ALPI P09923 1/20 0.38
ALPL P05186 1/20 0.36
MAOA P21397 6/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7388132 0.88 KCNH2 (0.40) HSD17B3MAOBIDO1KDM4EALDH1A1
SCHEMBL7383110 0.75 KCNH2 (0.38) HSD17B3MAOBIDO1KDM4EALDH1A1
SCHEMBL548396 0.73 IDO1 (0.45) HSD17B3MAOBIDO1KDM4EALDH1A1
SCHEMBL7495329 0.73 SLC6A4 (0.53) HSD17B3MAOBIDO1ACHEALPI
SCHEMBL7495322 0.73 SLC6A4 (0.53) HSD17B3MAOBIDO1ACHEALPI
SCHEMBL7450620 0.73 KDM4E (0.50) MAOBKDM4EALDH1A1
SCHEMBL8032293 0.72 MAOB (0.47) HSD17B3MAOBIDO1KDM4EALDH1A1
SCHEMBL18347517 0.71 IDO1 (0.51) HSD17B3MAOBIDO1KDM4EALDH1A1
SCHEMBL2256874 0.71 KDM4E (0.46) KDM4EALDH1A1GLAMAOA
SCHEMBL6635463 0.69 IDO1 (0.41) HSD17B3MAOBIDO1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0918768-B1 AROMATIC AMIDINE DERIVATIVES USEFUL AS SELECTIVE THROMBIN INHIBITORS C & C RES LAB (KR) 2002-01-09 EP disclosed
US-6201006-B1 ANTICOAGULANTS C & C RESEARCH LABORATORIES (KR) 2001-03-13 US disclosed
EP-0918768-A1 AROMATIC AMIDINE DERIVATIVES USEFUL AS SELECTIVE THROMBIN INHIBITORS C & C Research Laboratories (KR) 1999-06-02 EP disclosed
WO-1997045424-A1 AROMATIC AMIDINE DERIVATIVES USEFUL AS SELECTIVE THROMBIN INHIBITORS C & C RESEARCH LABORATORIES (KR) 1997-12-04 WO disclosed